SCHEMBL9535079

SCHEMBL9535079

Cc1nc2sccn2c(=O)c1CCN1CCC(Cc2nc3ccccc3n2Cc2ccco2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.45
ALDH1A1 P00352 5/20 0.45
MAPT P10636 4/20 0.45
HSD17B10 Q99714 3/20 0.45
CYP2D6 P10635 3/20 0.45
KDM4E B2RXH2 3/20 0.45
LMNA P02545 2/20 0.45
TP53 P04637 2/20 0.45
CYP2C9 P11712 2/20 0.45
ALOX15 P16050 2/20 0.45
DGKA P23743 2/20 0.45
TDP1 Q9NUW8 2/20 0.45
CYP2C19 P33261 1/20 0.45
HTR1A P08908 4/20 0.43
HTR2C P28335 3/20 0.43
HRH1 P35367 3/20 0.43
DRD2 P14416 3/20 0.43
HTR2A P28223 3/20 0.43
MEN1 O00255 2/20 0.43
CYP3A4 P08684 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9538894 0.89 SLC6A9 (0.44) TSHRALDH1A1MAPTHSD17B10CYP2D6
SCHEMBL8567881 0.89 MAPT (0.44) TSHRALDH1A1MAPTHSD17B10CYP2D6
SCHEMBL9536415 0.87 KDM4E (0.48) TSHRALDH1A1MAPTHSD17B10CYP2D6
SCHEMBL9536406 0.87 ALDH1A1 (0.37) TSHRALDH1A1HSD17B10KDM4ETDP1
SCHEMBL9537922 0.83 ALDH1A1 (0.38) TSHRALDH1A1MAPTHSD17B10KDM4E
SCHEMBL9537833 0.83 ALDH1A1 (0.39) TSHRALDH1A1HSD17B10KDM4ECYP2C9
SCHEMBL9536489 0.79 ADRA1A (0.48) TSHRALDH1A1MAPTHSD17B10CYP2D6
SCHEMBL9537953 0.78 KDM4E (0.46) TSHRALDH1A1MAPTHSD17B10CYP2D6
SCHEMBL9536136 0.77 SLC6A9 (0.44) TSHRALDH1A1HSD17B10KDM4ELMNA
Hydrochloric Acid SCHEMBL9535191 0.76 SLC6A9 (0.43) TSHRALDH1A1HSD17B10KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP claimed