SCHEMBL9536053

SCHEMBL9536053

CCc1onc(-c2c(F)cccc2Cl)c1OC(=O)Cl

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.53
SCN5A Q14524 1/20 0.53
SMN1; SMN2 Q16637 3/20 0.48
TP53 P04637 1/20 0.47
MAPT P10636 1/20 0.47
POLB P06746 2/20 0.47
KMT2A Q03164 2/20 0.46
ATM Q13315 1/20 0.46
LMNA P02545 2/20 0.46
ALDH1A1 P00352 3/20 0.45
GHSR Q92847 1/20 0.45
HPGD P15428 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
ALOX15 P16050 1/20 0.44
GPBAR1 Q8TDU6 1/20 0.44
NPC1 O15118 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9533421 0.92 SCN9A (0.49) SCN9ASCN5AMAPTPOLBKMT2A
SCHEMBL9537450 0.91 GHSR (0.47) SCN9ASCN5ASMN1; SMN2TP53MAPT
SCHEMBL9536365 0.84 LMNA (0.57) SCN9ASMN1; SMN2TP53MAPTPOLB
SCHEMBL9535220 0.82 GHSR (0.51) SCN9ASCN5AMAPTPOLBKMT2A
SCHEMBL9533125 0.81 KMT2A (0.48) SCN9ASMN1; SMN2POLBKMT2ALMNA
SCHEMBL9538504 0.81 GPBAR1 (0.53) SMN1; SMN2TP53MAPTPOLBLMNA
SCHEMBL9532926 0.76 PTGS1 (0.54) POLBKMT2ATSHRMAPK1ALOX15
SCHEMBL9538135 0.75 SMN1; SMN2 (0.48) SCN9ASCN5ASMN1; SMN2TP53MAPT
SCHEMBL9534075 0.75 SMN1; SMN2 (0.43) SCN9ASCN5ASMN1; SMN2TP53MAPT
SCHEMBL9535705 0.75 GPBAR1 (0.48) SMN1; SMN2GHSRGPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0573883-A1 Utilization of 3 substituted aryl-5-alkyl-isoxazole-4-carboxylic acid derivatives against endoparasites new 3-substituted aryl-5-alkyl-isoxazole-4-carboxylic acid derivatives and process for their preparation BAYER AG (DE) 1993-12-15 EP disclosed