SCHEMBL9536189

SCHEMBL9536189

Cc1ccc(Cc2ccnc(N)c2N)cc1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 5/20 0.47
NOS3 P29474 4/20 0.47
ROCK1 Q13464 1/20 0.40
NOS1 P29475 1/20 0.38
LTA4H P09960 1/20 0.38
IDO1 P14902 1/20 0.38
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5036404 0.84 NOS2 (0.46) NOS2NOS3ROCK1IDO1
SCHEMBL3906522 0.82 MPO (0.43) NOS2NOS3IDO1
SCHEMBL9694376 0.81 CYP17A1 (0.44) NOS2NOS3ROCK1ALDH1A1RAB9A
SCHEMBL7499087 0.81 LTA4H (0.43) NOS2NOS3ROCK1LTA4H
SCHEMBL9535888 0.81 ALDH1A1 (0.51) ROCK1LTA4HIDO1NPC1ALDH1A1
SCHEMBL5249618 0.79 MPO (0.46) LTA4HIDO1
SCHEMBL9390459 0.79 NOS3 (0.52) NOS2NOS3NOS1LTA4HNPC1
SCHEMBL22068695 0.78 NOS2 (0.47) NOS2NOS3NOS1ALDH1A1
SCHEMBL30612294 0.75 NOS3 (0.38) NOS2NOS3
SCHEMBL26921776 0.75 CHRNA1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed