SCHEMBL9537500

SCHEMBL9537500

CC(C)N1CCC(Cc2nc3cnccc3n2Cc2ccc(F)cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.46
ENPP2 Q13822 1/20 0.43
RAB9A P51151 1/20 0.42
CYP2D6 P10635 4/20 0.40
HRH1 P35367 4/20 0.40
CHRM1 P11229 2/20 0.40
HRH3 Q9Y5N1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9537449 0.84 SSTR5 (0.52) RAB9ACYP2D6HRH3
SCHEMBL10804293 0.81 KCNH2 (0.47) KCNH2RAB9ACYP2D6HRH1CHRM1
SCHEMBL10547773 0.80 HTR1A (0.56) KCNH2CYP2D6HRH1CHRM1HRH3
Oxalic Acid SCHEMBL9537077 0.76 HRH1 (0.56) KCNH2CYP2D6HRH1CHRM1HRH3
Oxalic Acid SCHEMBL9537074 0.76 HRH1 (0.56) KCNH2CYP2D6HRH1CHRM1HRH3
SCHEMBL9538842 0.76 SSTR5 (0.52) ENPP2RAB9ACYP2D6HRH3
SCHEMBL9537733 0.75 ENPP2 (0.44) ENPP2RAB9ACYP2D6HRH1
SCHEMBL9535904 0.75 KCNH2 (0.54) KCNH2ENPP2RAB9AHRH1CHRM1
SCHEMBL14507936 0.72 HRH3 (0.52) KCNH2HRH3
SCHEMBL9536543 0.72 SSTR5 (0.66) KCNH2RAB9ACYP2D6HRH1CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed
US-4839374-A TREATING ALLERGIES JANSSEN PHARMACEUTICA, N.V. (BE) 1989-06-13 US disclosed
EP-0151826-A1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1985-08-21 EP disclosed