SCHEMBL9537553

SCHEMBL9537553

CC(Cc1ccccn1)(OC(N)=O)C(=O)NC(CO)Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.43
CYP3A4 P08684 1/20 0.43
ROCK2 O75116 5/20 0.43
ROCK1 Q13464 5/20 0.43
RPS6KA5 O75582 1/20 0.43
RPS6KA4 O75676 1/20 0.43
PRKACA P17612 1/20 0.43
GSK3A P49840 1/20 0.43
GSK3B P49841 1/20 0.43
IRAK1 P51617 1/20 0.43
PRKX P51817 1/20 0.43
PRKG1 Q13976 1/20 0.43
PKN2 Q16513 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
SGK2 Q9HBY8 1/20 0.43
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 1/20 0.42
MAPT P10636 1/20 0.42
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7668995 0.80 MAPK1 (0.45) MAPK1CYP3A4ROCK2ROCK1RPS6KA5
SCHEMBL9700657 0.79 MMP8 (0.46) MAPK1CYP3A4CYP1A2MAPTSMN1; SMN2
SCHEMBL6888466 0.77 USP2 (0.47) MAPK1CYP3A4MAPTTSHRKMT2A
SCHEMBL9538634 0.76 MGLL (0.42) MAPK1CYP3A4ROCK2ROCK1RPS6KA5
SCHEMBL4339886 0.72 MAPK1 (0.63) MAPK1CYP3A4ROCK2ROCK1RPS6KA5
SCHEMBL9336196 0.71 KMT2A (0.47) MAPK1CYP3A4MAPTTSHRKMT2A
SCHEMBL4902230 0.71 ATM (0.48) CYP3A4CYP1A2ATM
SCHEMBL22559221 0.71 ATM (0.48) CYP3A4CYP1A2ATM
SCHEMBL4890941 0.71 ATM (0.48) CYP3A4CYP1A2ATM
SCHEMBL29638860 0.71 FDPS (0.46) MAPK1CYP1A2TSHRSMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993003721-A1 CHOLECYSTOKININ ANTAGONISTS USEFUL FOR TREATING DEPRESSION WARNER-LAMBERT COMPANY (US) 1993-03-04 WO claimed
WO-1993003721-A1 CHOLECYSTOKININ ANTAGONISTS USEFUL FOR TREATING DEPRESSION WARNER-LAMBERT COMPANY (US) 1993-03-04 WO disclosed