SCHEMBL9538008

SCHEMBL9538008

N#Cc1ccc(-c2occ3ccccc23)[nH]c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 1/20 0.42
KDM4E B2RXH2 7/20 0.41
ALDH1A1 P00352 6/20 0.41
GAA P10253 3/20 0.41
GLA P06280 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
MCL1 Q07820 2/20 0.36
HPGD P15428 3/20 0.36
HSD17B10 Q99714 1/20 0.36
PIM1 P11309 3/20 0.35
CLK1 P49759 1/20 0.34
DYRK1A Q13627 1/20 0.34
GALR3 O60755 1/20 0.34
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9754547 0.75 MCL1 (0.55) MDM2KDM4EALDH1A1GAAGLA
SCHEMBL9536884 0.74 KDM4E (0.46) MDM2KDM4EALDH1A1GAAGLA
SCHEMBL9535550 0.72 ALDH1A1 (0.53) MDM2KDM4EALDH1A1GAAGLA
SCHEMBL8123124 0.71 IMPDH2 (0.38) KDM4EALDH1A1CA1CA2MCL1
SCHEMBL4474609 0.71 MDM2 (0.62) MDM2KDM4EALDH1A1GAAGLA
SCHEMBL9536812 0.70 ALDH1A1 (0.60) MDM2KDM4EALDH1A1GAAGLA
SCHEMBL9538000 0.69 NPC1 (0.44) MDM2KDM4EALDH1A1GAAGLA
SCHEMBL9754436 0.69 ALDH1A1 (0.33) KDM4EALDH1A1HPGDHSD17B10NPC1
SCHEMBL9529006 0.69 MDM2 (0.47) MDM2KDM4EALDH1A1GAAGLA
SCHEMBL3836372 0.69 KDM4E (0.50) MDM2KDM4EALDH1A1GAAGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0532531-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1993-03-24 EP disclosed
WO-1991017987-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-11-28 WO disclosed