SCHEMBL9538770

SCHEMBL9538770

CC(C)(C)c1ccc(C=P(c2ccccc2)(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.41
ESRRG P62508 1/20 0.41
CYP1A2 P05177 1/20 0.39
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38
ALOX5 P09917 1/20 0.37
TSHR P16473 1/20 0.37
GRIN2D O15399 2/20 0.36
GRIN3B O60391 2/20 0.36
GRIN1 Q05586 2/20 0.36
GRIN2A Q12879 2/20 0.36
GRIN2B Q13224 2/20 0.36
GRIN2C Q14957 2/20 0.36
GRIN3A Q8TCU5 2/20 0.36
MAPT P10636 3/20 0.36
MEN1 O00255 1/20 0.36
MITF O75030 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9539528 0.81 ALDH1A1 (0.48) CYP1A2NR1H3TSHRKIF11RAB9A
SCHEMBL1132385 0.79 ALDH1A1 (0.39) CYP1A2ALOX5TSHRMAPTMEN1
SCHEMBL9538596 0.78 LMNA (0.42) TSHRMAPTHPGDSMN1; SMN2LMNA
SCHEMBL9539397 0.75 ALDH1A1 (0.41) CYP1A2MAPTSMN1; SMN2LMNATDP1
SCHEMBL24193844 0.74 ESR1 (0.50) MAPTMEN1GAAHPGDKMT2A
SCHEMBL9541503 0.74 TSHR (0.42) CYP1A2TSHRMAPTLMNA
SCHEMBL9541494 0.74 NFE2L2 (0.52) TSHRMAPTMEN1KMT2ASMN1; SMN2
SCHEMBL14269409 0.74 ALDH1A1 (0.42) MAPTMEN1GAAHPGDKMT2A
SCHEMBL7535089 0.73 CYP1A2 (0.55) TRPV1ESRRGCYP1A2NR1H2NR1H3
SCHEMBL6546384 0.73 CYP1A2 (0.55) TRPV1ESRRGCYP1A2NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0311955-B1 BICYCLIC PEROXIDE F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
US-4977184-A Bicyclic peroxides compositions for and treatment of malaria therewith HOFFMANN-LA ROCHE INC. (US) 1990-12-11 US disclosed
EP-0311955-A2 Bicyclic peroxide F. HOFFMANN-LA ROCHE AG (CH) 1989-04-19 EP disclosed