SCHEMBL9539397

SCHEMBL9539397

C(c1ccc(-c2ccccc2)cc1)=P(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
TP53 P04637 1/20 0.41
CA1 P00915 1/20 0.41
MGLL Q99685 1/20 0.41
HDAC2 Q92769 2/20 0.37
TAAR1 Q96RJ0 3/20 0.37
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
MAPK1 P28482 2/20 0.37
HSD17B10 Q99714 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MMP3 P08254 1/20 0.37
BCL2L1 Q07817 1/20 0.37
MAPT P10636 2/20 0.36
LMNA P02545 1/20 0.36
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.34
SIRT1 Q96EB6 1/20 0.34
SIRT3 Q9NTG7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1132385 0.85 ALDH1A1 (0.39) ALDH1A1CA1HDAC2CYP1A2MAPK1
Fluoride SCHEMBL27260416 0.83 ALDH1A1 (0.38) ALDH1A1CA1HDAC2CYP1A2MAPK1
SCHEMBL10744618 0.83 TP53 (0.43) TP53TAAR1TDP1MAPTLMNA
SCHEMBL9541494 0.80 NFE2L2 (0.52) ALDH1A1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL9541503 0.80 TSHR (0.42) CYP1A2HSD17B10MAPTLMNASIRT1
SCHEMBL24193844 0.80 ESR1 (0.50) ALDH1A1CA1TAAR1CYP3A4TDP1
SCHEMBL9538596 0.80 LMNA (0.42) ALDH1A1CYP3A4TDP1MAPTLMNA
SCHEMBL14269409 0.80 ALDH1A1 (0.42) ALDH1A1MAPK1TDP1MAPTLMNA
SCHEMBL14423637 0.77 LTA4H (0.48) ALDH1A1CA1LMNAL3MBTL1NPC1
Benzaldehyde SCHEMBL6051056 0.76 ALDH1A1 (0.61) ALDH1A1MAPK1HSD17B10TDP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0311955-B1 BICYCLIC PEROXIDE F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
US-5134240-A Malaria therapy HOFFMANN-LAROCHE, INC. (US) 1992-07-28 US disclosed
US-4977184-A Bicyclic peroxides compositions for and treatment of malaria therewith HOFFMANN-LA ROCHE INC. (US) 1990-12-11 US disclosed
EP-0311955-A2 Bicyclic peroxide F. HOFFMANN-LA ROCHE AG (CH) 1989-04-19 EP disclosed