SCHEMBL9539333

SCHEMBL9539333

CCN(C(=O)c1ccc(CBr)cc1)[C@@](CC)(CCC(=O)O)C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.34
PPARG P37231 1/20 0.34
ALDH1A1 P00352 6/20 0.33
ALDH2 P05091 1/20 0.33
MAPT P10636 2/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
RAB9A P51151 1/20 0.33
HDAC6 Q9UBN7 2/20 0.32
HDAC1 Q13547 1/20 0.32
HPGD P15428 3/20 0.32
HSD17B10 Q99714 1/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
THRB P10828 1/20 0.32
KMT2A Q03164 1/20 0.32
NR1H4 Q96RI1 1/20 0.32
MLYCD O95822 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10758621 0.90 L3MBTL1 (0.38) L3MBTL1PPARGALDH1A1ALDH2LMNA
SCHEMBL6308181 0.85 TPMT (0.34) L3MBTL1PPARGALDH1A1MAPTLMNA
SCHEMBL6311889 0.85 ALDH1A1 (0.36) ALDH1A1MAPTNPC1LMNARAB9A
SCHEMBL10965940 0.84 ALDH1A1 (0.38) ALDH1A1MAPTNPC1RAB9AHPGD
SCHEMBL6648900 0.82 HPGD (0.34) ALDH1A1MAPTRAB9AHDAC1HPGD
SCHEMBL10828836 0.77 OPRD1 (0.33) HPGD
SCHEMBL9556353 0.77 LMNA (0.43) ALDH1A1MAPTNPC1LMNARAB9A
SCHEMBL7666244 0.76
SCHEMBL6655035 0.74 MEN1 (0.37) ALDH1A1MEN1CYP1A2THRBKMT2A
SCHEMBL11712059 0.72 HPGD (0.43) CES2CES1LMNAHDAC6HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0215063-B1 PYRIDO (2,3-d )PYRIMIDIN DERIVATIVES UNIV PRINCETON (US) 1993-11-03 EP disclosed
US-5026851-A Antineoplastic agents THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-06-25 US disclosed
US-4845216-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1989-07-04 US disclosed
EP-0215063-A4 PYRIDO (2,3-d )PYRIMIDIN DERIVATIVES. UNIV PRINCETON (US) 1987-11-23 EP disclosed
EP-0215063-A1 PYRIDO (2,3-d )PYRIMIDIN DERIVATIVES. UNIV PRINCETON (US) 1987-03-25 EP disclosed
WO-1986005181-A1 PYRIDO AD2,3-d BDPYRIMIDIN DERIVATIVES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1986-09-12 WO disclosed