SCHEMBL9539807

SCHEMBL9539807

C[C@H]1CNc2c(cccc2[N+](=O)[O-])CN1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PNMT P11086 5/20 0.43
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
ACHE P22303 1/20 0.39
TDP1 Q9NUW8 2/20 0.39
TSHR P16473 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PDE10A Q9Y233 1/20 0.36
GPR35 Q9HC97 1/20 0.35
POLB P06746 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP3A4 P08684 1/20 0.35
ALOX15 P16050 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9539813 1.00 PNMT (0.43) PNMTADRA2AADRA2BADRA2CCHRNB2
SCHEMBL7903541 0.78 TDP1 (0.40) PNMTADRA2AADRA2BADRA2CCHRNB2
SCHEMBL27453650 0.78 PNMT (0.41) PNMTADRA2AADRA2BADRA2CTSHR
SCHEMBL16269182 0.77 PNMT (0.55) PNMTADRA2AADRA2BADRA2CCHRNB2
SCHEMBL9701418 0.75 CHRNB2 (0.40) PNMTCHRNB2CHRNA4ACHETDP1
SCHEMBL7480596 0.75 TDP1 (0.38) PNMTADRA2AADRA2BADRA2CTDP1
SCHEMBL7903560 0.74 TDP1 (0.39) CHRNB2CHRNA4TDP1TSHRSMN1; SMN2
SCHEMBL7903558 0.74 TDP1 (0.39) CHRNB2CHRNA4TDP1TSHRSMN1; SMN2
SCHEMBL7903563 0.74 TDP1 (0.39) CHRNB2CHRNA4TDP1TSHRSMN1; SMN2
SCHEMBL7391102 0.74 CD44 (0.34) PNMTADRA2AADRA2BADRA2CALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0557307-A1 PROCESS FOR PRODUCING 4,5,6,7-TETRAHYDRO-IMIDAZO-(4,5,LJK) (1,4)-BENZODIAZEPINE-2-(1H)-THIONES AND INTERMEDIATE PRODUCTS Roche Diagnostics GmbH (DE) 1993-09-01 EP disclosed
WO-1992008706-A1 PROCESS FOR PRODUCING 4,5,6,7-TETRAHYDRO-IMIDAZO-(4,5,LJK) (1,4)-BENZODIAZEPINE-2-(1H)-THIONES AND INTERMEDIATE PRODUCTS BOEHRINGER MANNHEIM GMBH (DE) 1992-05-29 WO disclosed