SCHEMBL9542741

SCHEMBL9542741

COc1cccc(CCN(CC(=O)N2Cc3ccccc3C[C@@H]2CC(=O)O)C(=O)[C@H]2Cc3ccccc3N2C(=O)OC(C)(C)C)c1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.37
OXTR P30559 1/20 0.36
AVPR1A P37288 1/20 0.36
NR1D1 P20393 1/20 0.36
OPRM1 P35372 1/20 0.36
HDAC8 Q9BY41 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9543510 0.93 ALDH1A1 (0.43) OXTRAVPR1AHDAC8ALDH1A1
SCHEMBL9543406 0.93 PTPN1 (0.38) HDAC8
SCHEMBL9543619 0.91 DRD2 (0.38) CFTRHDAC8
SCHEMBL9542649 0.89 PREP (0.39) HDAC8
SCHEMBL9543607 0.88 ALDH1A1 (0.39) ALDH1A1MAPT
SCHEMBL9544819 0.88 DRD4 (0.38)
SCHEMBL9545071 0.87 DRD2 (0.37) OXTRAVPR1AOPRM1MAPT
SCHEMBL9544446 0.86 HDAC8 (0.36) OPRM1HDAC8
SCHEMBL9542714 0.86 PREP (0.41) HDAC8
SCHEMBL9543221 0.85 DRD2 (0.35) OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993020099-A2 CCK AND/OR GASTRIN RECEPTOR LIGANDS FERRING B.V. (NL) 1993-10-14 WO claimed
WO-1993020099-A2 CCK AND/OR GASTRIN RECEPTOR LIGANDS FERRING B.V. (NL) 1993-10-14 WO disclosed