SCHEMBL9542935

SCHEMBL9542935

c1ccc(-n2ccc3ncnc-3n2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.43
CYP2C9 P11712 1/20 0.41
MAPT P10636 3/20 0.39
TSHR P16473 2/20 0.39
HSD17B10 Q99714 2/20 0.39
ADORA2A P29274 1/20 0.39
ADORA2B P29275 1/20 0.39
ADORA1 P30542 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PDE10A Q9Y233 1/20 0.39
HPGD P15428 1/20 0.38
LMNA P02545 2/20 0.38
ALDH1A1 P00352 3/20 0.38
NOTUM Q6P988 1/20 0.37
GAA P10253 1/20 0.36
GRM5 P41594 2/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 1/20 0.36
EGFR P00533 1/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10691844 0.73 SMN1; SMN2 (0.45) MAPTTSHRADORA2AADORA2BADORA1
SCHEMBL218118 0.72 KMT2A (0.57) HTTCYP2C9MAPTTSHRHSD17B10
SCHEMBL12854024 0.71 HTT (0.50) HTTCYP2C9MAPTTSHRHSD17B10
Ammonia Solution, Strong SCHEMBL10418488 0.71 KMT2A (0.55) HTTCYP2C9MAPTTSHRHSD17B10
SCHEMBL2148390 0.70 ALDH1A1 (0.46) HTTCYP2C9HSD17B10L3MBTL1HPGD
SCHEMBL3923785 0.70 GRM5 (0.64) HTTCYP2C9MAPTTSHRHSD17B10
SCHEMBL30795324 0.70 GRM5 (0.64) HTTCYP2C9MAPTTSHRHSD17B10
SCHEMBL3648026 0.70 RXRA (0.36) CYP2C9GRM5CYP1A2CYP2C19
SCHEMBL7844771 0.69 HTT (0.56) HTTCYP2C9HSD17B10L3MBTL1PDE10A
SCHEMBL10689031 0.69 KDM4E (0.50) MAPTTSHRHSD17B10ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993003033-A1 CARBONATE-SUBSTITUTED IMIDAZO[4,5-d] PYRIDAZINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G. D. SEARLE & CO. (US) 1993-02-18 WO disclosed
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed
WO-1991019715-A1 1H-SUBSTITUTED-IMIDAZO[4,5-d]PYRIDAZINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1991-12-26 WO disclosed
US-4722929-A Novel 2-phenyl-imidazoles and pharmaceutical compositions containing same DR. KARL THOMAE GMBH (DE) 1988-02-02 US disclosed
EP-0149200-A1 Novel 2-pnenyl-imidazoles, their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1985-07-24 EP disclosed