SCHEMBL9543549

SCHEMBL9543549

Fc1cc(C2CCC(/C=C/Cl)CC2)ccc1C(F)(F)F.Fc1cc(C2CCC(/C=C/Cl)CC2)ccc1OC(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.39
HTR2A P28223 1/20 0.33
EPHX2 P34913 4/20 0.32
PDE2A O00408 5/20 0.32
RXRA P19793 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2B Q13224 1/20 0.31
PTK2 Q05397 1/20 0.30
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963026 0.93 EPHX2 (0.36) KDM1AEPHX2PDE2A
SCHEMBL8963018 0.93 EPHX2 (0.36) KDM1AEPHX2PDE2A
SCHEMBL8962943 0.90 EPHX2 (0.34) EPHX2PDE2A
SCHEMBL8962822 0.89 KDM1A (0.47) KDM1AHTR2APDE2ARXRAGRIN1
SCHEMBL8962830 0.89 KDM1A (0.47) KDM1AHTR2APDE2ARXRAGRIN1
SCHEMBL8962898 0.86 KDM1A (0.43) KDM1AHTR2APDE2ARXRAGRIN1
SCHEMBL8963179 0.84 CTSK (0.37) EPHX2PDE2AGRIN2B
SCHEMBL8963176 0.84 CTSK (0.37) EPHX2PDE2AGRIN2B
SCHEMBL12997536 0.80 EPHX2 (0.45) KDM1AEPHX2PDE2A
SCHEMBL8963103 0.80 KIF11 (0.46) KDM1ACYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993007234-A1 HALOVINYL-DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-15 WO disclosed