SCHEMBL8963103

SCHEMBL8963103

Fc1cc(-c2ccc([C@H]3CC[C@H](/C=C/Cl)CC3)cc2)ccc1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 12/20 0.46
CYP11B2 P19099 7/20 0.43
CYP11B1 P15538 6/20 0.43
KDM1A O60341 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963089 1.00 KIF11 (0.46) KIF11CYP11B2CYP11B1KDM1A
SCHEMBL8962822 0.89 KDM1A (0.47) KIF11CYP11B2CYP11B1KDM1A
SCHEMBL8962830 0.89 KDM1A (0.47) KIF11CYP11B2CYP11B1KDM1A
SCHEMBL8962898 0.86 KDM1A (0.43) KIF11CYP11B2CYP11B1KDM1A
SCHEMBL8963237 0.85 P2RY14 (0.35) CYP11B2CYP11B1KDM1A
SCHEMBL8963228 0.85 P2RY14 (0.35) CYP11B2CYP11B1KDM1A
SCHEMBL8962836 0.83 JAK2 (0.35) CYP11B2CYP11B1
SCHEMBL8962842 0.83 JAK2 (0.35) CYP11B2CYP11B1
SCHEMBL8962838 0.82 SLC6A3 (0.39)
SCHEMBL8962923 0.82 KDM1A (0.37) KIF11KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed
WO-1993007234-A1 HALOVINYL-DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-15 WO disclosed