SCHEMBL954665

SCHEMBL954665

CCCCC(=O)Nc1cc(-c2nnn[nH]2)ccc1F

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
GSK3A P49840 1/20 0.40
SOAT1 P35610 2/20 0.39
RORC P51449 2/20 0.39
CETP P11597 1/20 0.39
POLB P06746 1/20 0.39
ADORA1 P30542 1/20 0.39
PARP1 P09874 1/20 0.39
CCNT1 O60563 1/20 0.39
CDK9 P50750 1/20 0.39
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20777935 0.84 SOAT1 (0.46) ALDH1A1SOAT1TP53MAPT
SCHEMBL20777938 0.82 ALDH1A1 (0.48) ALDH1A1SOAT1TP53MAPT
SCHEMBL956335 0.79 HPGD (0.60) KDM4EALDH1A1GSK3ALMNATP53
SCHEMBL20777974 0.79 RAB9A (0.51) KDM4EALDH1A1SOAT1POLBLMNA
SCHEMBL28569542 0.79 RAB9A (0.51) KDM4EALDH1A1SOAT1POLBLMNA
SCHEMBL949484 0.78 SMN1; SMN2 (0.42) KDM4EALDH1A1GSK3ARORCADORA1
SCHEMBL1309175 0.77 ALDH1A1 (0.58) KDM4EALDH1A1POLB
SCHEMBL20777929 0.73 PSMB11 (0.62) ALDH1A1SOAT1POLBLMNATP53
SCHEMBL26318663 0.72 SOAT2 (0.58) KDM4EALDH1A1SOAT1POLBLMNA
SCHEMBL23412427 0.72 KDM4E (0.50) KDM4EALDH1A1SOAT1CETPPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011006935-A2 TETRAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed