SCHEMBL9555151

SCHEMBL9555151

CCOC(=O)CCNC(=O)CCCCNC(=O)OC(C)(C)C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.53
TDP1 Q9NUW8 1/20 0.51
CYP3A4 P08684 2/20 0.47
CA1 P00915 4/20 0.47
CA2 P00918 4/20 0.47
CA12 O43570 2/20 0.47
CA9 Q16790 2/20 0.47
CTSK P43235 1/20 0.47
MAOA P21397 1/20 0.46
MAOB P27338 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25827510 0.96 GAA (0.54) GAATDP1CYP3A4CA1CA2
SCHEMBL15728746 0.91 CTSK (0.50) GAATDP1CA1CA2CA12
SCHEMBL25095054 0.90 TDP1 (0.58) GAATDP1CYP3A4CA1CA2
SCHEMBL8032622 0.89 GAA (0.69) GAATDP1CYP3A4CA1CA2
SCHEMBL5653695 0.88 TDP1 (0.61) GAATDP1CYP3A4CA1CA2
SCHEMBL7158127 0.88 TDP1 (0.61) GAATDP1CYP3A4CA1CA2
SCHEMBL29256392 0.88 TDP1 (0.61) GAATDP1CYP3A4CA1CA2
SCHEMBL1784924 0.88 CTSK (0.51) GAATDP1CA1CA2CA12
SCHEMBL7405019 0.86 GAA (0.64) GAATDP1CYP3A4CA1CA2
SCHEMBL23782441 0.86 MAOA (0.55) GAATDP1CYP3A4CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5250517-A Hypotensive and cardiotonic agents; cardiac insufficiency HOFFMANN-LA ROCHE INC. (US) 1993-10-05 US disclosed