SCHEMBL9558246

SCHEMBL9558246

COc1cc2ccc(C(=O)CCCCCBr)cc2cc1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.50
ALDH1A1 P00352 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2C19 P33261 1/20 0.50
HSD17B10 Q99714 1/20 0.50
HDAC1 Q13547 5/20 0.48
HDAC8 Q9BY41 3/20 0.48
CTNNB1 P35222 2/20 0.48
WNT3A P56704 2/20 0.48
THRA P10827 1/20 0.43
THRB P10828 1/20 0.43
PDE4B Q07343 2/20 0.43
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PTPN1 P18031 1/20 0.43
HTR1A P08908 1/20 0.43
XDH P47989 1/20 0.43
PDE4A P27815 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9557967 0.99 HPGD (0.51) HPGDALDH1A1CYP1A2CYP2C19HSD17B10
SCHEMBL6344166 0.89 THRA (0.55) HPGDALDH1A1CYP1A2CYP2C19HSD17B10
SCHEMBL6340900 0.89 THRA (0.55) HPGDALDH1A1CYP1A2CYP2C19HSD17B10
SCHEMBL27200216 0.87 CTNNB1 (0.63) ALDH1A1CYP1A2CYP2C19CTNNB1WNT3A
SCHEMBL5355533 0.87 CTNNB1 (0.63) ALDH1A1CYP1A2CYP2C19CTNNB1WNT3A
SCHEMBL9119840 0.85 CTNNB1 (0.65) ALDH1A1CYP1A2CYP2C19CTNNB1WNT3A
SCHEMBL6348421 0.84 HPGD (0.51) HPGDALDH1A1CYP1A2CYP2C19HSD17B10
SCHEMBL6543390 0.83 PTPN1 (0.62) HPGDALDH1A1CYP1A2CYP2C19HSD17B10
SCHEMBL30682871 0.81 HPGD (0.75) HPGDALDH1A1CYP1A2CYP2C19HSD17B10
SCHEMBL9558005 0.81 ALDH1A1 (0.54) HPGDALDH1A1CYP1A2CYP2C19HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0384350-B1 DIHYDROXY NAPHTHALENE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-28 EP disclosed
EP-0384350-A1 Dihydroxy naphthalene derivatives F. HOFFMANN-LA ROCHE AG (CH) 1990-08-29 EP disclosed
US-4937371-A INHIBITING LIPOXYGENASE HOFFMANN-LA ROCHE INC. (US) 1990-06-26 US disclosed