SCHEMBL9558248

SCHEMBL9558248

CC(C)(C)OC(=O)N1CCN(CCOC(=O)N[C@@H](Cc2ccccc2)C(=O)O)CC1

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.58
ITGB3 P05106 3/20 0.56
ITGA2B P08514 3/20 0.56
YAP1 P46937 1/20 0.54
P2RX7 Q99572 8/20 0.53
HRH2 P25021 1/20 0.53
HRH1 P35367 1/20 0.53
ACE P12821 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27841545 0.90 ITGB3 (0.53) MAPK1ITGB3ITGA2BYAP1P2RX7
SCHEMBL9558243 0.87 YAP1 (0.64) MAPK1YAP1P2RX7ACE
SCHEMBL7276592 0.85 POLB (0.65) MAPK1YAP1ACE
SCHEMBL7276597 0.85 POLB (0.65) MAPK1YAP1ACE
SCHEMBL6349585 0.82 P2RX7 (0.73) MAPK1YAP1P2RX7
SCHEMBL27841549 0.82 YAP1 (0.52) ITGB3ITGA2BYAP1P2RX7HRH2
SCHEMBL27841551 0.82 YAP1 (0.52) ITGB3ITGA2BYAP1P2RX7HRH2
SCHEMBL6165579 0.80 MAPK1 (0.75) MAPK1YAP1
SCHEMBL6165580 0.80 MAPK1 (0.75) MAPK1YAP1
SCHEMBL9558236 0.80 MAPK1 (0.64) MAPK1YAP1ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5215968-A Hypotension agents and viricides HOECHST AKTIENGESELLSCHAFT (DE) 1993-06-01 US disclosed
EP-0373497-A2 Dipeptide derivatives with an enzyme-inhibiting activity HOECHST AKTIENGESELLSCHAFT (DE) 1990-06-20 EP disclosed