SCHEMBL9564461

SCHEMBL9564461

CN1CCN(c2nc3c(c(N)c2N)c(=O)cc(C(=O)O)n3C2CC2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.37
CDK1 P06493 1/20 0.37
AURKB Q96GD4 1/20 0.37
ALDH1A1 P00352 8/20 0.36
CYP1A2 P05177 8/20 0.36
USP2 O75604 7/20 0.36
CASP1 P29466 7/20 0.36
CASP7 P55210 7/20 0.36
HSD17B10 Q99714 6/20 0.36
CYP2C9 P11712 4/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
HIF1A Q16665 3/20 0.36
GLA P06280 2/20 0.36
TSHR P16473 2/20 0.36
MAPK1 P28482 2/20 0.35
CYP2D6 P10635 1/20 0.35
PIM1 P11309 1/20 0.35
PIM3 Q86V86 1/20 0.35
PIM2 Q9P1W9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564483 0.83 PIK3CA (0.37) AURKACDK1AURKBALDH1A1CYP1A2
SCHEMBL9564474 0.77 KDM4E (0.39) ALDH1A1CYP1A2USP2CASP1CASP7
SCHEMBL9564467 0.70 KDM4E (0.41) ALDH1A1HSD17B10MEN1KMT2ATSHR
SCHEMBL9564504 0.70 RXFP1 (0.42) ALDH1A1MEN1KMT2A
SCHEMBL9088365 0.69 MAPKAPK3 (0.44) AURKBPIM1PIM3PIM2TOP2A
Hydrochloric Acid SCHEMBL9564479 0.67 SCN5A (0.34) ALDH1A1CYP1A2USP2CASP1CASP7
SCHEMBL9805870 0.66 CNR1 (0.47) CNR2
SCHEMBL9564459 0.64 MEN1 (0.40) ALDH1A1CYP1A2USP2CASP1CASP7
SCHEMBL8741056 0.64 TOP2A (0.40) MAPK1TOP2ATOP2B
SCHEMBL6801320 0.63 ALDH1A1 (0.40) ALDH1A1CYP1A2USP2CASP1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0531958-A1 6-Aminoquinolones, their synthesis and their use as antibacterial agents MEDIOLANUM FARMACEUTICI S.P.A. (IT) 1993-03-17 EP disclosed