SCHEMBL9564483

SCHEMBL9564483

CN1CCN(c2nc3c(cc2N)c(=O)cc(C(=O)O)n3C2CC2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 5/20 0.37
AURKA O14965 1/20 0.37
CDK1 P06493 1/20 0.37
AURKB Q96GD4 1/20 0.37
HRH4 Q9H3N8 4/20 0.37
ALDH1A1 P00352 4/20 0.36
CYP1A2 P05177 4/20 0.36
HSD17B10 Q99714 4/20 0.36
USP2 O75604 3/20 0.36
CASP1 P29466 3/20 0.36
CASP7 P55210 3/20 0.36
EEF2K O00418 3/20 0.36
MAPK1 P28482 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 2/20 0.35
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35
EEF2 P13639 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564504 0.86 RXFP1 (0.42) PIK3CAALDH1A1EEF2KMEN1KMT2A
SCHEMBL9564461 0.83 AURKA (0.37) AURKACDK1AURKBHRH4ALDH1A1
SCHEMBL9564467 0.79 KDM4E (0.41) ALDH1A1HSD17B10MAPK1MEN1KMT2A
Hydrochloric Acid SCHEMBL9564479 0.76 SCN5A (0.34) ALDH1A1CYP1A2HSD17B10USP2CASP1
SCHEMBL9805870 0.73 CNR1 (0.47) PIK3CAEEF2KEEF2CNR2
SCHEMBL9564472 0.68 KDM4E (0.42) AURKAAURKBALDH1A1CYP1A2HSD17B10
SCHEMBL7094750 0.68 DPP4 (0.39) HSD17B10KMT2A
SCHEMBL9564474 0.68 KDM4E (0.39) ALDH1A1CYP1A2HSD17B10USP2CASP1
SCHEMBL6801320 0.67 ALDH1A1 (0.40) HRH4ALDH1A1CYP1A2HSD17B10USP2
SCHEMBL10877952 0.67 ADH5 (0.38) CYP1A2HSD17B10USP2MAPK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0531958-A1 6-Aminoquinolones, their synthesis and their use as antibacterial agents MEDIOLANUM FARMACEUTICI S.P.A. (IT) 1993-03-17 EP disclosed