SCHEMBL9564803

SCHEMBL9564803

CCOC(=O)N1CCC(Nc2nc3cncnc3n2Cc2cnccn2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 5/20 0.46
NOS1 P29475 4/20 0.44
NOS3 P29474 2/20 0.44
ALDH1A1 P00352 5/20 0.44
HSD17B10 Q99714 4/20 0.44
HPGD P15428 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
MAP4K4 O95819 1/20 0.43
KDM4E B2RXH2 4/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
MAPT P10636 2/20 0.41
TSHR P16473 2/20 0.41
LMNA P02545 2/20 0.41
NR2F2 P24468 1/20 0.41
HTT P42858 1/20 0.41
CDK1 P06493 3/20 0.40
CDK4 P11802 3/20 0.40
CCND1 P24385 3/20 0.40
CDK2 P24941 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9602879 0.90 NOS2 (0.56) NOS2NOS1NOS3ALDH1A1HSD17B10
SCHEMBL9564948 0.86 ALDH1A1 (0.42) NOS2NOS1NOS3ALDH1A1HSD17B10
SCHEMBL9564864 0.85 ALDH1A1 (0.51) NOS2NOS1NOS3ALDH1A1HSD17B10
SCHEMBL9564853 0.84 ALDH1A1 (0.52) NOS2NOS1NOS3ALDH1A1HSD17B10
Bromide SCHEMBL10428854 0.83 NOS2 (0.52) NOS2NOS1NOS3ALDH1A1HSD17B10
SCHEMBL9564902 0.83 USP2 (0.51) NOS2NOS1NOS3ALDH1A1HSD17B10
Bromide SCHEMBL9698287 0.83 NOS2 (0.51) NOS2NOS1NOS3ALDH1A1HSD17B10
SCHEMBL9565029 0.83 ALDH1A1 (0.51) NOS2NOS1NOS3ALDH1A1HSD17B10
SCHEMBL9564774 0.83 ALDH1A1 (0.44) NOS2NOS1NOS3ALDH1A1HSD17B10
SCHEMBL9564839 0.82 NOS2 (0.50) NOS2NOS1NOS3ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
EP-0206415-B1 (4-PIPERIDINYLMETHYL AND -HETERO)PURINES JANSSEN PHARMACEUTICA N.V. (BE) 1993-01-27 EP disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed