SCHEMBL9564853

SCHEMBL9564853

CCOC(=O)N1CCC(Nc2nc3cncnc3n2Cc2ccc(C)cc2C)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
LMNA P02545 2/20 0.52
MAPT P10636 2/20 0.52
TSHR P16473 2/20 0.52
NR2F2 P24468 1/20 0.52
HTT P42858 1/20 0.52
NOS2 P35228 5/20 0.48
NOS1 P29475 4/20 0.48
NOS3 P29474 2/20 0.48
MAP4K4 O95819 1/20 0.45
HSD17B10 Q99714 3/20 0.44
HPGD P15428 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
KDM4E B2RXH2 3/20 0.43
CDK1 P06493 2/20 0.41
CDK4 P11802 2/20 0.41
CCND1 P24385 2/20 0.41
CDK2 P24941 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564864 0.84 ALDH1A1 (0.51) ALDH1A1SMN1; SMN2LMNAMAPTTSHR
SCHEMBL9564803 0.84 NOS2 (0.46) ALDH1A1SMN1; SMN2LMNAMAPTTSHR
SCHEMBL9564902 0.83 USP2 (0.51) ALDH1A1SMN1; SMN2LMNAMAPTTSHR
SCHEMBL9564774 0.82 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2LMNAMAPTTSHR
SCHEMBL9565029 0.82 ALDH1A1 (0.51) ALDH1A1SMN1; SMN2LMNAMAPTHTT
SCHEMBL9602879 0.82 NOS2 (0.56) ALDH1A1SMN1; SMN2MAPTTSHRNOS2
SCHEMBL9564950 0.82 SOS1 (0.42) ALDH1A1LMNAHSD17B10
SCHEMBL9564849 0.82 SMN1; SMN2 (0.50) ALDH1A1SMN1; SMN2LMNAMAPTTSHR
SCHEMBL9564816 0.82 NOS2 (0.46) ALDH1A1SMN1; SMN2LMNAMAPTTSHR
SCHEMBL9564948 0.81 ALDH1A1 (0.42) ALDH1A1SMN1; SMN2LMNAMAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
EP-0206415-B1 (4-PIPERIDINYLMETHYL AND -HETERO)PURINES JANSSEN PHARMACEUTICA N.V. (BE) 1993-01-27 EP disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed