SCHEMBL9565029

SCHEMBL9565029

CCOC(=O)N1CCC(Nc2nc3cncnc3n2Cc2ccc(OC)cc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.51
LMNA P02545 3/20 0.51
GAA P10253 2/20 0.51
NOS2 P35228 5/20 0.49
NOS1 P29475 4/20 0.49
NOS3 P29474 2/20 0.49
HSD17B10 Q99714 3/20 0.46
HPGD P15428 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
SSTR5 P35346 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
MAPT P10636 3/20 0.45
PDE5A O76074 2/20 0.45
POLB P06746 1/20 0.45
MAPK1 P28482 1/20 0.45
MAP4K4 O95819 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
USP2 O75604 2/20 0.44
KDM4E B2RXH2 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564902 0.91 USP2 (0.51) ALDH1A1LMNAGAANOS2NOS1
SCHEMBL9564864 0.91 ALDH1A1 (0.51) ALDH1A1LMNANOS2NOS1NOS3
SCHEMBL9629419 0.88 USP2 (0.48) ALDH1A1LMNAGAANOS2NOS1
SCHEMBL9602879 0.83 NOS2 (0.56) ALDH1A1NOS2NOS1NOS3HSD17B10
SCHEMBL9564774 0.83 ALDH1A1 (0.44) ALDH1A1LMNANOS2NOS1NOS3
SCHEMBL9564803 0.83 NOS2 (0.46) ALDH1A1LMNANOS2NOS1NOS3
SCHEMBL9698901 0.82 LMNA (0.73) ALDH1A1LMNAGAANOS2NOS1
SCHEMBL9564853 0.82 ALDH1A1 (0.52) ALDH1A1LMNANOS2NOS1NOS3
SCHEMBL9564816 0.82 NOS2 (0.46) ALDH1A1LMNANOS2NOS1NOS3
SCHEMBL9564849 0.82 SMN1; SMN2 (0.50) ALDH1A1LMNANOS2NOS1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
EP-0206415-B1 (4-PIPERIDINYLMETHYL AND -HETERO)PURINES JANSSEN PHARMACEUTICA N.V. (BE) 1993-01-27 EP disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed