SCHEMBL9564863

SCHEMBL9564863

Oc1ccc(CCN2CCC(Cc3nc4c(O)ncnc4n3Cc3ccc(F)cc3)CC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.48
KCNH2 Q12809 1/20 0.48
SSTR5 P35346 1/20 0.40
GRIN2B Q13224 2/20 0.40
GRIN1 Q05586 1/20 0.40
NPY1R P25929 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564878 0.91 HRH1 (0.49) KCNH2SSTR5
SCHEMBL9564783 0.87 CYP3A4 (0.39) KCNH2
SCHEMBL10547724 0.82 SLC6A9 (0.55) NR4A2KCNH2SSTR5
Bromide SCHEMBL9564766 0.81 KCNH2 (0.42) NR4A2KCNH2
SCHEMBL9565008 0.80 DRD2 (0.50) KCNH2
SCHEMBL9539974 0.79 KCNH2 (0.69) NR4A2KCNH2SSTR5
SCHEMBL10553768 0.79 KCNH2 (0.57) NR4A2KCNH2SSTR5GRIN2BGRIN1
SCHEMBL9564927 0.79 P2RX7 (0.44) KCNH2
Water SCHEMBL9536552 0.78 KCNH2 (0.56) NR4A2KCNH2SSTR5GRIN2BGRIN1
SCHEMBL9564825 0.78 HTR1A (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed