SCHEMBL9564876

SCHEMBL9564876

CCOC(=O)N1CCC(Cc2nc3c(Cl)ncnc3n2Cc2ccc(F)cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.46
CASP1 P29466 1/20 0.46
CASP7 P55210 1/20 0.46
GAA P10253 3/20 0.42
GRIN2B Q13224 2/20 0.41
ALDH1A1 P00352 5/20 0.40
HPGD P15428 4/20 0.40
LMNA P02545 3/20 0.40
KDM4E B2RXH2 3/20 0.40
HTT P42858 2/20 0.40
PIK3CD O00329 1/20 0.40
TP53 P04637 1/20 0.40
TRPC3 Q13507 1/20 0.40
TRPC7 Q9HCX4 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MAPT P10636 4/20 0.39
OPRD1 P41143 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564912 0.92 HSD17B10 (0.46) HSD17B10CASP1CASP7GAAGRIN2B
SCHEMBL9564937 0.86 HSD17B10 (0.47) HSD17B10CASP1CASP7GAAGRIN2B
SCHEMBL9564964 0.80 ALDH1A1 (0.46) ALDH1A1LMNA
SCHEMBL9564783 0.76 CYP3A4 (0.39) HSD17B10CASP1CASP7ALDH1A1TSHR
SCHEMBL10550194 0.75 KCNH2 (0.46) HSD17B10CASP1CASP7GAAALDH1A1
SCHEMBL10553680 0.75 KCNH2 (0.46) HSD17B10CASP1CASP7GAAALDH1A1
SCHEMBL9564841 0.73 USP2 (0.49) HSD17B10CASP1CASP7GAAALDH1A1
SCHEMBL9866073 0.73 CCR3 (0.44) ALDH1A1LMNATSHR
SCHEMBL9564786 0.73 ALDH1A1 (0.47) HSD17B10CASP1CASP7GAAALDH1A1
SCHEMBL9564830 0.71 SSTR5 (0.43) LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
EP-0206415-B1 (4-PIPERIDINYLMETHYL AND -HETERO)PURINES JANSSEN PHARMACEUTICA N.V. (BE) 1993-01-27 EP disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed