SCHEMBL9564890

SCHEMBL9564890

Fc1ccc(Cn2c(CC3CCN(Cc4ccccc4)CC3)nc3ncnc(Cl)c32)cc1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
CCR3 P51677 1/20 0.45
SSTR5 P35346 1/20 0.45
SLC6A4 P31645 2/20 0.44
SLC6A3 Q01959 2/20 0.44
TSHR P16473 1/20 0.43
BCHE P06276 1/20 0.43
ACHE P22303 1/20 0.43
BACE1 P56817 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564964 0.84 ALDH1A1 (0.46) ALDH1A1CCR3SSTR5SLC6A4SLC6A3
SCHEMBL9564865 0.82 SSTR5 (0.63) SSTR5SLC6A4SLC6A3BCHEACHE
SCHEMBL9536547 0.81 SSTR5 (0.52) ALDH1A1CCR3SSTR5SLC6A4SLC6A3
SCHEMBL9564937 0.80 HSD17B10 (0.47) ALDH1A1TSHR
SCHEMBL9866073 0.78 CCR3 (0.44) ALDH1A1CCR3SSTR5SLC6A4SLC6A3
SCHEMBL9536543 0.77 SSTR5 (0.66) ALDH1A1SSTR5SLC6A3TSHR
SCHEMBL9564956 0.77 CYP1A2 (0.54) ALDH1A1CCR3SSTR5TSHR
SCHEMBL9535367 0.76 SLC6A9 (0.58) CCR3SSTR5
SCHEMBL9564830 0.76 SSTR5 (0.43) CCR3SSTR5ACHEBACE1
SCHEMBL9565004 0.73 HTR1A (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed