SCHEMBL9567458

SCHEMBL9567458

COc1cnccc1N1CCN(CCCc2c[nH]c3ccccc23)C(C)C1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 8/20 0.49
HTR7 P34969 3/20 0.47
SLC6A4 P31645 1/20 0.47
KCNH2 Q12809 1/20 0.47
MEN1 O00255 1/20 0.46
LMNA P02545 1/20 0.46
KMT2A Q03164 1/20 0.46
DRD2 P14416 5/20 0.45
HTR2A P28223 2/20 0.44
HTR6 P50406 2/20 0.44
SSTR4 P31391 1/20 0.41
SSTR3 P32745 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9262251 0.99 HTR1A (0.48) HTR1AHTR7SLC6A4KCNH2MEN1
SCHEMBL9567460 0.85 HTR1A (0.63) HTR1AHTR7SLC6A4KCNH2DRD2
Hydrochloric Acid SCHEMBL9264804 0.84 HTR1A (0.65) HTR1AHTR7SLC6A4KCNH2DRD2
SCHEMBL6362332 0.79 DRD2 (0.44) HTR1AHTR7SLC6A4KCNH2DRD2
SCHEMBL9204485 0.78 LMNA (0.46) HTR1AHTR7MEN1LMNAKMT2A
SCHEMBL6362295 0.77 HTR1A (0.55) HTR1AHTR7SLC6A4KCNH2DRD2
SCHEMBL19431749 0.76 HTR1A (0.65) HTR1AHTR7SLC6A4KMT2ADRD2
SCHEMBL6356579 0.75 HTR1A (0.47) HTR1AHTR7SLC6A4KCNH2MEN1
SCHEMBL9208142 0.75 HTR1A (0.48) HTR1ASLC6A4DRD2
SCHEMBL6356825 0.74 HTR1A (0.53) HTR1AHTR7SLC6A4KCNH2HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0548813-A1 Antimigraine 4-pyrimidinyl and pyridinyl derivatives of indol-3yl-alkyl piperazines Bristol-Myers Squibb Company (US) 1993-06-30 EP claimed