SCHEMBL9569322

SCHEMBL9569322

COc1ccc(-c2cn3c(n2)sc2ccccc23)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 6/20 0.73
MAPT P10636 4/20 0.73
RAB9A P51151 3/20 0.73
LMNA P02545 2/20 0.73
SMN1; SMN2 Q16637 2/20 0.73
TSHR P16473 1/20 0.73
ATM Q13315 1/20 0.73
TDP1 Q9NUW8 1/20 0.73
APP P05067 1/20 0.63
RXFP1 Q9HBX9 1/20 0.59
THRB P10828 2/20 0.57
ALDH1A1 P00352 2/20 0.55
NPC1 O15118 2/20 0.55
GAA P10253 1/20 0.55
NFKB1 P19838 1/20 0.55
GFER P55789 1/20 0.55
NFKB2 Q00653 1/20 0.55
RELA Q04206 1/20 0.55
KDM4E B2RXH2 2/20 0.53
POLB P06746 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11015064 0.87 TP53 (0.73) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL11012567 0.85 TP53 (0.57) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL13650900 0.85 LMNA (0.55) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL11015014 0.84 TP53 (1.00) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL11015020 0.84 TP53 (0.81) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL84416 0.84 RAB9A (0.64) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL24106015 0.83 TP53 (0.55) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL11351985 0.83 MAPT (0.61) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL13198300 0.82 TP53 (0.70) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL10803793 0.82 TP53 (0.60) TP53MAPTRAB9ALMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11559518-B2 Endoplasmic reticulum stress regulator comprising benzothiazoimidazolyl compound ER STRESS RESEARCH INSTITUTE, INC. (JP) 2023-01-24 US disclosed
US-20210386715-A1 ENDOPLASMIC RETICULUM STRESS REGULATOR COMPRISING BENZOTHIAZOIMIDAZOLYL COMPOUND ER STRESS RESEARCH INSTITUTE, INC. (JP) 2021-12-16 US disclosed
EP-0524055-A1 Imidazo(2,1-b)benzothiazole-3-acetamide derivatives, process for their preparation and their therapeutical use SYNTHELABO (FR) 1993-01-20 EP disclosed
US-4497817-A ANTIALLERGENS-IMMUNOSUPPRESSIVE AGENTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1985-02-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11559518-B2 Endoplasmic reticulum stress regulator comprising benzothiazoimidazolyl compound HSPA5, DNAJC10, ERP44 TP53 1281/4885MAPT 3116/4885RAB9A 1684/4885
US-20210386715-A1 ENDOPLASMIC RETICULUM STRESS REGULATOR COMPRISING BENZOTHIAZOIMIDAZOLYL COMPOUND DNAJC10, HSPA5, ERP44 TP53 1668/4885MAPT 3271/4885RAB9A 2027/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.