SCHEMBL9577811

SCHEMBL9577811

Oc1ccc(N=C2NCCN2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S100B P04271 1/20 0.39
CA12 O43570 3/20 0.38
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
CA9 Q16790 3/20 0.38
MEN1 O00255 2/20 0.38
NPC1 O15118 2/20 0.38
KMT2A Q03164 2/20 0.38
ESR1 P03372 4/20 0.37
ESR2 Q92731 4/20 0.37
GLB1 P16278 1/20 0.37
CTRB1 P17538 1/20 0.37
CTRC Q99895 1/20 0.37
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
GMNN O75496 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
CA3 P07451 1/20 0.36
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10974740 0.98 CA12 (0.40) S100BCA12CA1CA2CA9
SCHEMBL3782607 0.77 HPGD (0.42) MEN1NPC1KMT2AMAPTKDM4E
SCHEMBL11215407 0.77 MAPT (0.44) CA12CA2CA9MEN1NPC1
SCHEMBL9421173 0.77 PTGS1 (0.37) CA1CA2MEN1KMT2AMAPT
SCHEMBL1741629 0.76 ALDH1A1 (0.39) MEN1NPC1KMT2AMAPTKDM4E
Hydrochloric Acid SCHEMBL10815621 0.76 MAPT (0.42) CA12CA2CA9MEN1NPC1
Bromide SCHEMBL11354612 0.76 BACE1 (0.35)
Bromide SCHEMBL11356265 0.74 SELL (0.31)
SCHEMBL10969178 0.72 ALDH1A1 (0.38) CA12CA1CA2CA9MEN1
SCHEMBL10967741 0.72 ALOX15 (0.41) MEN1KMT2AMAPTKDM4ECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5180721-A Imidazoline substituted naphthalene compounds for treatment of glaucoma ALLERGAN, INC. (US) 1993-01-19 US claimed
WO-1992021349-A1 COMBINATIONS OF ALPHA-2 ADRENERGIC AGONISTS WITH ALPHA-3 ANTAGONISTS FOR LOWERING INTRAOCULAR PRESSURE ALLERGAN, INC. (US) 1992-12-10 WO claimed
EP-0399791-A1 Combinations of selective alpha-adrenergic agonists and antagonists useful in lowering intraocular pressure ALLERGAN, INC (US) 1990-11-28 EP claimed
EP-0086126-B1 IMIDAZOLINE DERIVATIVES, THEIR PREPARATION AND THERAPEUTICAL APPLICATION SYNTHELABO (FR) 1985-07-24 EP claimed
US-4492709-A VISION DEFECTX SYNTHELABO (FR) 1985-01-08 US disclosed