SCHEMBL9585437

SCHEMBL9585437

COc1ccc(-c2c(O)c(C(=O)O)c(C)c3cc(O)ccc23)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.51
MEN1 O00255 5/20 0.44
KMT2A Q03164 5/20 0.44
ESRRA P11474 1/20 0.44
MAPT P10636 5/20 0.42
LMNA P02545 1/20 0.42
HPGD P15428 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
HTT P42858 2/20 0.42
HSD17B10 Q99714 2/20 0.42
PKM P14618 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
HIF1A Q16665 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
TP53 P04637 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303055 0.85 ERAP1 (0.48) MEN1KMT2AMAPTLMNAHPGD
SCHEMBL9391003 0.78 GPR35 (0.40) CSNK2A2CSNK2BESR2KDM4E
SCHEMBL9270518 0.77 LDHA (0.40) NPC1KMT2ATSHRCYP3A4CYP2C9
SCHEMBL9898347 0.71 DHODH (0.50) LMNAHPGDHSD17B10TSHRCYP2C9
SCHEMBL28664927 0.71 LDHA (0.49) MAPTLMNAHPGDSMN1; SMN2HTT
SCHEMBL6652685 0.71 KDM4E (0.49) NPC1MEN1KMT2AMAPTLMNA
SCHEMBL8353016 0.69 SMN1; SMN2 (0.59) HPGDSMN1; SMN2HSD17B10CYP2C9CYP2C19
SCHEMBL11253942 0.68 HPGD (0.51) NPC1MEN1KMT2AESRRAMAPT
SCHEMBL6383991 0.68 SMN1; SMN2 (0.54) NPC1MAPTLMNAHPGDSMN1; SMN2
SCHEMBL5427914 0.68 NPC1 (1.00) NPC1MEN1KMT2AMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5227399-A Pyranylphenyl naphthalene lactones as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA, INC. (CA) 1993-07-13 US disclosed
EP-0501579-A1 Naphthalene lactones as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA INC. (CA) 1992-09-02 EP disclosed