SCHEMBL9593284

SCHEMBL9593284

CN1C(=O)CC(C)(C)c2cc(N)ccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.46
HDAC1 Q13547 2/20 0.45
HDAC6 Q9UBN7 2/20 0.45
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC9 Q9UKV0 1/20 0.45
ATAD2 Q6PL18 1/20 0.38
BACE1 P56817 5/20 0.37
FSHR P23945 1/20 0.36
RARA P10276 1/20 0.36
RARB P10826 1/20 0.36
RARG P13631 1/20 0.36
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
RXRA P19793 2/20 0.35
KMT2A Q03164 2/20 0.34
KDM4E B2RXH2 2/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2060570 0.84 ATAD2 (0.39) CYP19A1HDAC1HDAC6HDAC3HDAC4
SCHEMBL20335480 0.81 ATAD2 (0.43) CYP19A1HDAC1HDAC6HDAC3HDAC4
SCHEMBL5736954 0.81 HDAC1 (0.47) HDAC1HDAC6HDAC3HDAC4HDAC2
SCHEMBL8310907 0.80 ATAD2 (0.55) CYP19A1HDAC1HDAC6ATAD2RXRA
SCHEMBL7709931 0.80 RARA (0.56) CYP19A1HDAC1HDAC6ATAD2FSHR
SCHEMBL6073600 0.78 LMNA (0.51) HDAC1HDAC6HDAC3HDAC4HDAC2
SCHEMBL9593368 0.78 ALDH1A1 (0.51) HDAC1HDAC6HDAC3HDAC4HDAC2
SCHEMBL6770006 0.77 HDAC1 (0.56) HDAC1HDAC6HDAC3HDAC4HDAC2
SCHEMBL9593493 0.77 HDAC1 (0.56) HDAC1HDAC6HDAC3HDAC4HDAC2
SCHEMBL6748962 0.76 NOTUM (0.45) HDAC1HDAC6HDAC3HDAC4HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5216148-A Treating, preventing neoplasms, dermatoses, aging of skin HOFFMANN-LA ROCHE INC. (US) 1993-06-01 US disclosed
EP-0504695-A1 New carboxamides, their preparation and pharmaceutical compositions containing them F. HOFFMANN-LA ROCHE AG (CH) 1992-09-23 EP disclosed