SCHEMBL9601090

SCHEMBL9601090

Cc1c(N2CCN(CCCC(c3ccc(F)cc3)c3ccc(F)cc3)CC2)nc(F)c(F)c1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 2/20 0.48
FAAH O00519 1/20 0.48
TSHR P16473 1/20 0.48
ALOX12 P18054 1/20 0.48
MAPK1 P28482 1/20 0.48
MTOR P42345 1/20 0.48
RAB9A P51151 1/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
DRD3 P35462 6/20 0.47
DRD2 P14416 5/20 0.47
HTR2A P28223 4/20 0.47
ADRA1A P35348 4/20 0.47
HRH1 P35367 4/20 0.47
OPRK1 P41145 4/20 0.47
SLC6A3 Q01959 4/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9602632 0.90 MEN1 (0.49) CYP3A4CYP2D6FAAHTSHRALOX12
SCHEMBL12786020 0.76 DRD3 (0.48) CYP3A4CYP2D6FAAHTSHRALOX12
SCHEMBL9602299 0.75 HTR2A (0.52) CYP3A4CYP2D6FAAHTSHRALOX12
SCHEMBL28876807 0.75 CYP3A4 (0.64) CYP3A4CYP2D6FAAHTSHRALOX12
SCHEMBL9516792 0.73 CYP3A4 (0.63) CYP3A4CYP2D6FAAHTSHRALOX12
SCHEMBL9602967 0.73 SIGMAR1 (0.79) DRD2CYP1A2CYP2C9SIGMAR1KDM4E
SCHEMBL9601301 0.73 DRD2 (0.56) CYP3A4CYP2D6FAAHTSHRALOX12
SCHEMBL9601882 0.73 SIGMAR1 (0.56) CYP3A4CYP2D6FAAHTSHRALOX12
SCHEMBL9602079 0.73 SLC6A9 (0.55) CYP3A4CYP2D6FAAHTSHRALOX12
Hydrochloric Acid SCHEMBL9603075 0.72 SLC6A2 (0.64) DRD3DRD2HTR2AHRH1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308476-B1 BISPHENYLALKYLPIPERAZINE DERIVATIVES, A METHOD OF THEIR PREPARATION AND A PHARMACEUTICAL PREPARATION Kabi Pharmacia AB (SE) 1993-02-03 EP disclosed
US-4937245-A ANTIDEPRESSANTS, ANXIOLYTIC AGENTS FEX TOMAS (SE) 1990-06-26 US disclosed