SCHEMBL9602856

SCHEMBL9602856

CC(O[Si](C)(C)C(C)(C)C)c1ccncc1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
CYP19A1 P11511 4/20 0.36
CYP17A1 P05093 3/20 0.36
GAA P10253 1/20 0.34
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
APLNR P35414 2/20 0.31
KIF11 P52732 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9185287 0.82 ADRA2B (0.38) SLC6A4SLC6A3
SCHEMBL26125646 0.79 NPC1 (0.33) APLNR
SCHEMBL31042359 0.79 APLNR (0.42) CYP3A4APLNR
SCHEMBL21556841 0.79 APLNR (0.31) APLNR
SCHEMBL31073192 0.79 APLNR (0.42) CYP3A4APLNR
SCHEMBL26125642 0.79 NPC1 (0.33) APLNR
SCHEMBL7196103 0.79 APLNR (0.31) APLNR
SCHEMBL408604 0.79 APLNR (0.42) CYP3A4APLNR
SCHEMBL17362036 0.77 KIF11 (0.31) KIF11
SCHEMBL18056394 0.77 CA2 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5217963-A Antiischemic, antiepileptic agent CIBA-GEIGY CORPORATION (US) 1993-06-08 US disclosed
US-5057506-A Anticonvulsants, antispasmodic and antischemic agents CIBA-GEIGY CORPORATION (US) 1991-10-15 US disclosed
US-4906621-A Certain 2-carboxypiperidyl-alkylene phosphonic acids and esters thereof useful for the treatment of disorders responsive to N-methyl-D-aspartate receptor blockade CIBA-GEIGY CORPORATION (US) 1990-03-06 US disclosed