SCHEMBL9603417

SCHEMBL9603417

COc1ccc2c(c1)S(=O)(=O)NC(C(=O)O)=N2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.46
CA9 Q16790 4/20 0.46
CA12 O43570 3/20 0.46
CA1 P00915 3/20 0.46
CA7 P43166 2/20 0.46
CA4 P22748 1/20 0.46
ABCC8 Q09428 1/20 0.40
KCNJ11 Q14654 1/20 0.40
KDM4E B2RXH2 3/20 0.40
MAPT P10636 2/20 0.40
POLB P06746 2/20 0.40
KMT2A Q03164 1/20 0.40
SLC40A1 Q9NP59 2/20 0.39
ALPI P09923 2/20 0.38
NFKBIA P25963 2/20 0.38
RELA Q04206 2/20 0.38
ALPL P05186 2/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
RECQL P46063 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20777878 0.83 ALDH1A1 (0.43) CA2CA9CA12CA1CA7
SCHEMBL20777832 0.79 KMT2A (0.39) POLBKMT2A
SCHEMBL20777728 0.78 CA2 (0.36) CA2CA9CA12CA1CA7
SCHEMBL20777563 0.70 ELANE (0.40) KDM4EMAPTPOLBSLC40A1ALDH1A1
SCHEMBL9606078 0.70 CHEK1 (0.44) CA2CA9CA12CA1CA7
SCHEMBL9604292 0.70 CA2 (0.36) CA2CA9CA12CA1CA7
SCHEMBL20777795 0.69 CFTR (0.43) CA2CA1KDM4EMAPTSLC40A1
SCHEMBL5186168 0.68 CA12 (0.63) CA2CA9CA12CA1CA7
SCHEMBL6720672 0.67 PTGES (0.57) CA2CA9CA12CA1CA7
SCHEMBL20773655 0.66 GABRA2 (0.43) CA2CA9CA12CA1CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993021171-A1 USE OF 2H-1,2,4-BENZOTHIADIAZINE-1,1-DIOXIDE-3-CARBOXYLIC ACID DERIVATIVES FOR PREPARING NMDA/AMPA RECEPTOR ANTAGONIST DRUGS, NOVEL PRODUCTS, PREPARATION THEREOF AND DRUGS CONTAINING SAME RHONE-POULENC RORER S.A. (FR) 1993-10-28 WO disclosed