SCHEMBL9608978

SCHEMBL9608978

CCc1c(F)ccc(C)c1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.41
CD38 P28907 1/20 0.35
PKM P14618 1/20 0.35
TAAR1 Q96RJ0 1/20 0.31
NOS3 P29474 1/20 0.31
NOS2 P35228 1/20 0.31
ALDH1A1 P00352 2/20 0.31
CYP3A4 P08684 1/20 0.31
ALOX15 P16050 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
ACHE P22303 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
FPR3 P25089 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL91338 0.84 P2RX7 (0.37) P2RX7CD38PKMTAAR1ALDH1A1
SCHEMBL11891675 0.81 NOS3 (0.40) P2RX7NOS3NOS2ALDH1A1CYP3A4
SCHEMBL488564 0.81 P2RX7 (0.40) P2RX7CD38PKMTAAR1CYP3A4
SCHEMBL1167603 0.81 P2RX7 (0.43) P2RX7CD38PKMTAAR1ALDH1A1
SCHEMBL146651 0.81 P2RX7 (0.40) P2RX7CD38PKMTAAR1CYP3A4
SCHEMBL856367 0.81 P2RX7 (0.40) P2RX7CD38PKMTAAR1ALDH1A1
SCHEMBL4120436 0.80 TAAR1 (0.36) P2RX7CD38PKMTAAR1ALDH1A1
SCHEMBL11888502 0.79 TAAR1 (0.50) P2RX7CD38TAAR1CYP1A2
SCHEMBL20326196 0.78 CYP3A4 (0.39) CYP3A4ALOX15SMN1; SMN2MEN1KMT2A
SCHEMBL21567308 0.77 ALDH1A1 (0.39) NOS3NOS2ALDH1A1CYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120135975-A1 Substituted Esters as Cannabinoid-1 Receptor Modulators MERCK & CO., INC. (US) 2012-05-31 US disclosed
US-20120071461-A1 Substituted Benzamide Compounds GRUENENTHAL GMBH (DE) 2012-03-22 US disclosed
US-20080312435-A1 Imine Compound TAISHO PHARMACEUTICAL CO., LTD. (JP) 2008-12-18 US disclosed
US-7279484-B2 Suppress tumor necrosis factor; Crohn's disease; imflammatory bowel disorders; sepsis; autoimmune disease AJINOMOTO CO., INC. (JP) 2007-10-09 US disclosed
US-7279484-B2 Suppress tumor necrosis factor; Crohn's disease; imflammatory bowel disorders; sepsis; autoimmune disease AJINOMOTO CO., INC. (JP) 2007-10-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080312435-A1 Imine Compound CNR1, CNR2, HRH4 P2RX7 225/4885CD38 659/4885PKM 3896/4885
US-20120135975-A1 Substituted Esters as Cannabinoid-1 Receptor Modulators CNR1, CNR2, FAAH P2RX7 1478/4885CD38 933/4885PKM 3476/4885
US-20120071461-A1 Substituted Benzamide Compounds BDKRB1, BDKRB2, HRH2 P2RX7 140/4885CD38 540/4885PKM 1255/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.