Olmesartan Medoxomil

Olmesartan Medoxomil

SCHEMBL96150

CCCc1nc(C(C)(C)O)c(C(=O)OCc2oc(=O)oc2C)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.79

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

AGTR1

The experimentally established mechanism targets of Olmesartan Medoxomil. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AGTR1 known ✓ P30556 11/20 0.79
AGTR2 P50052 12/20 0.79
ABCC3 O15438 1/20 0.79
ABCC4 O15439 1/20 0.79
ABCB11 O95342 1/20 0.79
CYP3A4 P08684 1/20 0.79
PDE4D Q08499 1/20 0.79
PDE3A Q14432 1/20 0.79
SLCO1B3 Q9NPD5 1/20 0.79
TDP1 Q9NUW8 1/20 0.79
SLCO1B1 Q9Y6L6 1/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2844872 0.96 AGTR2 (0.73) AGTR2AGTR1ABCC3ABCC4ABCB11
SCHEMBL15132375 0.95 AGTR2 (0.72) AGTR2AGTR1ABCC3ABCC4ABCB11
SCHEMBL6857515 0.95 AGTR2 (0.71) AGTR2AGTR1ABCC3ABCC4ABCB11
SCHEMBL7302860 0.94 AGTR2 (0.71) AGTR2AGTR1ABCC3ABCC4ABCB11
SCHEMBL4019176 0.94 AGTR1 (0.70) AGTR2AGTR1ABCC3ABCC4ABCB11
SCHEMBL2626709 0.93 AGTR2 (0.69) AGTR2AGTR1ABCC3ABCC4ABCB11
SCHEMBL6434240 0.93 AGTR2 (0.70) AGTR2AGTR1ABCC3ABCC4ABCB11
SCHEMBL7886557 0.93 AGTR2 (0.68) AGTR2AGTR1ABCC3ABCC4ABCB11
SCHEMBL7883447 0.93 AGTR2 (0.68) AGTR2AGTR1ABCC3ABCC4ABCB11
SCHEMBL8243357 0.91 AGTR2 (0.65) AGTR2AGTR1ABCC3ABCC4ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 249 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230321046-A1 PHARMACEUTICAL COMPOSITION OF SINGLE DOSAGE FORM FOR TREATING OR PREVENTING HYPERTENSION AND HYPERLIPIDEMIA DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2023-10-12 US claimed
EP-4205730-A1 PHARMACEUTICAL COMPOSITION OF SINGLE DOSAGE FORM FOR TREATING OR PREVENTING HYPERTENSION AND HYPERLIPIDEMIA Daewoong Pharmaceutical Co., Ltd. (KR) 2023-07-05 EP claimed
EP-3045174-A1 MEDICINE FOR PREVENTION OF AND TREATMENT FOR ARTERIOSCLEROSIS AND HYPERTENSION Daiichi Sankyo Company, Limited (JP) 2016-07-20 EP claimed
EP-2517728-B1 Olmesartan medoxomil for preventing or treating angiogenic eye diseases DAIICHI SANKYO CO LTD (JP) 2015-01-28 EP claimed
EP-2174666-B1 MEDICINAL AGENT FOR TREATMENT OF AMYLOID BETA-INDUCED CEREBRAL CIRCULATION OR CEREBRAL BLOOD FLOW DISORDERS DAIICHI SANKYO CO LTD (JP) 2013-12-18 EP claimed
US-20120302614-A1 METHOD FOR IMPROVING CEREBRAL CIRCULATION OR TREATING A CEREBRAL BLOOD FLOW DISORDER OSAKA UNIVERSITY (JP) 2012-11-29 US claimed
EP-2517728-A1 Drug for preventing or treating angiogenic eye diseases Daiichi Sankyo Company, Limited (JP) 2012-10-31 EP claimed
EP-2334668-A1 PROCESS FOR PREPARING OLMESARTAN MEDOXOMIL INTERMEDIATE Krka Tovarna Zdravil, D.D., Novo Mesto (SI) 2011-06-22 EP claimed
US-20100130567-A1 MEDICAL AGENT FOR PREVENTION OR TREATMENT OF ALZHEIMER 'S DISEASE DAIICHI SANKYO COMPANY, LIMITED (JP) 2010-05-27 US claimed
EP-2174666-A1 MEDICINAL AGENT FOR PREVENTION OR TREATMENT OF ALZHEIMER'S DISEASE Daiichi Sankyo Company, Limited (JP) 2010-04-14 EP claimed
EP-1872783-A1 THERAPEUTIC AGENT FOR CORNEAL/CONJUNCTIVAL DISORDER SANTEN PHARMACEUTICAL CO., LTD. (JP) 2008-01-02 EP claimed
US-20070203211-A1 Drug for preventing or treating angiogenic eye diseases SANKYO COMPANY, LIMITED (JP) 2007-08-30 US claimed
US-20060252806-A1 synergistic use of angiotensin II receptor antagonist like (5-methyl-2-oxo-1,3-dioxolen-4-yl)methyl 4-(1-hydroxy-1-methylethyl)-2-propyl-1-[[2'-(1H-tetrazol-5-yl)biphenyl-4-yl]methyl]imidazol-5-carboxylate with the calcium channel blockers; calcium channel blockers containing 1,4-dihydropyridine group SANKYO COMPANY LIMITED (JP) 2006-11-09 US claimed
US-20060252805-A1 Medicine for prevention of and treatment for arteriosclerosis and hypertension SANKYO COMPANY LIMITED (JP) 2006-11-09 US claimed
US-20060009502-A1 Medicine for prevention of and treatment for arteriosclerosis and hypertension SANKYO COMPANY, LIMITED (JP) 2006-01-12 US claimed
EP-1614428-A1 DRUG FOR PREVENTING OR TREATING ANGIOGENIC EYE DISEASES Sankyo Company, Limited (JP) 2006-01-11 EP claimed
EP-1604664-A1 MEDICINE FOR PREVENTION OF AND TREATMENT FOR ARTERIOSCLEROSIS AND HYPERTENSION Sankyo Company, Limited (JP) 2005-12-14 EP claimed
EP-0503785-B1 1-Biphenylimidazole derivatives, their preparation and their therapeutic use SANKYO CO (JP) 2001-04-25 EP claimed
US-5616599-A HYPOTENSIVE AGENTS FOR CARDIOVASCULAR DISORDER SANKYO COMPANY, LIMITED (JP) 1997-04-01 US claimed
EP-0503785-A1 1-Biphenylimidazole derivatives, their preparation and their therapeutic use Sankyo Company Limited (JP) 1992-09-16 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100130567-A1 MEDICAL AGENT FOR PREVENTION OR TREATMENT OF ALZHEIMER 'S DISEASE AGTR1, AGTR2, ACE AGTR1 1/4885AGTR2 2/4885ABCC3 1034/4885
US-20060252805-A1 Medicine for prevention of and treatment for arteriosclerosis and hypertension AGTR1, AGTR2, EDNRB AGTR1 1/4885AGTR2 2/4885ABCC3 754/4885
US-20120302614-A1 METHOD FOR IMPROVING CEREBRAL CIRCULATION OR TREATING A CEREBRAL BLOOD FLOW DISORDER AGTR2, AGTR1, BDKRB2 AGTR1 2/4885AGTR2 1/4885ABCC3 1984/4885
US-20060252806-A1 synergistic use of angiotensin II receptor antagonist like (5-methyl-2-oxo-1,3-dioxolen-4-yl)methyl 4-(1-hydroxy-1-methylethyl)-2-propyl-1-[[2'-(1H-tetrazol-5-yl)biphenyl-4-yl]methyl]imidazol-5-carboxylate with the calcium channel blockers; calcium channel blockers containing 1,4-dihydropyridine group AGTR1, AGTR2, CACNA1D AGTR1 1/4885AGTR2 2/4885ABCC3 2182/4885
US-20060009502-A1 Medicine for prevention of and treatment for arteriosclerosis and hypertension AGTR2, AGTR1, REN AGTR1 2/4885AGTR2 1/4885ABCC3 1064/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.