SCHEMBL9622705

SCHEMBL9622705

C[S+]([O-])CCOc1cc(N)c(Cl)cc1C(=O)NCC1(O)CN2CCC1CC2

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.44
HTR3A P46098 5/20 0.42
HTR3E A5X5Y0 3/20 0.42
HTR3B O95264 3/20 0.42
HTR3D Q70Z44 3/20 0.42
HTR3C Q8WXA8 3/20 0.42
HTR5A P47898 1/20 0.42
MEN1 O00255 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
HTR4 Q13639 1/20 0.41
DRD4 P21917 2/20 0.41
DRD3 P35462 2/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9623046 0.89 HTR3A (0.47) DRD2HTR3AHTR3EHTR3BHTR3D
SCHEMBL9623235 0.87 DRD2 (0.45) DRD2HTR3AHTR3EHTR3BHTR3D
SCHEMBL9622424 0.85 HTR3A (0.58) DRD2HTR3AHTR3EHTR3BHTR3D
SCHEMBL9474052 0.84 HTR3E (0.46) DRD2HTR3AHTR3EHTR3BHTR3D
Fumaric Acid SCHEMBL9622753 0.84 CYP3A4 (0.46) DRD2HTR3AHTR3EHTR3BHTR3D
Fumaric Acid SCHEMBL9622764 0.84 CYP3A4 (0.46) DRD2HTR3AHTR3EHTR3BHTR3D
SCHEMBL9623137 0.83 DRD2 (0.44) DRD2HTR3AHTR3EHTR3BHTR3D
SCHEMBL9622432 0.82 DRD2 (0.49) DRD2HTR3AHTR3EHTR3BHTR3D
SCHEMBL9622821 0.79 HTR4 (0.40) DRD2HTR3AHTR3EHTR3BHTR3D
SCHEMBL9623047 0.79 MEN1 (0.42) DRD2HTR3AHTR3EHTR3BHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5137895-A Antiemetic, anxiolytic, gastric emptying and serotonin modulating activity A. H. ROBINS COMPANY, INCORPORATED (US) 1992-08-11 US disclosed