SCHEMBL9623047

SCHEMBL9623047

Nc1cc(OCC2CCCCO2)c(C(=O)NCC2(O)CN3CCC2CC3)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
KMT2A Q03164 2/20 0.42
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
HTR1A P08908 1/20 0.42
ADRA2A P08913 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
ADRA2B P18089 1/20 0.42
HTR2C P28335 1/20 0.42
SLC6A4 P31645 1/20 0.42
DRD3 P35462 1/20 0.42
HTR2B P41595 1/20 0.42
KCNH2 Q12809 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
DRD2 P14416 2/20 0.42
HTR3A P46098 5/20 0.41
HTR3E A5X5Y0 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9623046 0.82 HTR3A (0.47) MEN1CYP2C9CYP2C19KMT2ADRD3
SCHEMBL9622424 0.81 HTR3A (0.58) MEN1CYP2C9CYP2C19KMT2ADRD2
SCHEMBL9623137 0.81 DRD2 (0.44) MEN1CYP2C9CYP2C19KMT2ADRD2
SCHEMBL9623235 0.79 DRD2 (0.45) MEN1CYP2C9CYP2C19KMT2ADRD3
SCHEMBL9622705 0.79 DRD2 (0.44) MEN1CYP2C9CYP2C19KMT2ADRD3
SCHEMBL9622432 0.78 DRD2 (0.49) MEN1CYP2C9CYP2C19KMT2ALMNA
SCHEMBL9622821 0.77 HTR4 (0.40) MEN1CYP2C9CYP2C19KMT2ADRD3
SCHEMBL9622761 0.77 PRKAB2 (0.43) KMT2AHTR4
Fumaric Acid SCHEMBL9622753 0.77 CYP3A4 (0.46) MEN1CYP2C9CYP2C19KMT2ACYP3A4
Fumaric Acid SCHEMBL9622764 0.77 CYP3A4 (0.46) MEN1CYP2C9CYP2C19KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5137895-A Antiemetic, anxiolytic, gastric emptying and serotonin modulating activity A. H. ROBINS COMPANY, INCORPORATED (US) 1992-08-11 US disclosed