SCHEMBL9623229

SCHEMBL9623229

COc1ccc(Oc2cc3c(c4c2[nH]c2ccc(OCc5ccccc5)cc24)C(=O)N(CCN(C)C)C3=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 2/20 0.44
SLC6A4 P31645 1/20 0.41
HTR1D P28221 1/20 0.41
TRPM8 Q7Z2W7 1/20 0.41
CCNE2 O96020 1/20 0.41
CDK4 P11802 1/20 0.41
PRKACA P17612 1/20 0.41
PRKACG P22612 1/20 0.41
PRKACB P22694 1/20 0.41
CCND1 P24385 1/20 0.41
CCNE1 P24864 1/20 0.41
CDK2 P24941 1/20 0.41
MAOA P21397 2/20 0.39
MAOB P27338 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MYLK Q15746 1/20 0.39
ROCK2 O75116 1/20 0.38
PLK1 P53350 1/20 0.38
CTSV O60911 2/20 0.38
CTSL P07711 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9622462 0.90 CHEK1 (0.45) CHEK1SLC6A4HTR1DTRPM8CCNE2
SCHEMBL9623319 0.87 ROCK2 (0.48) CHEK1CDK4CCND1MYLKROCK2
Hydrochloric Acid SCHEMBL9622616 0.86 ROCK2 (0.47) CHEK1CDK4CCND1MYLKROCK2
SCHEMBL9623280 0.85 KDM4E (0.45) CHEK1HTR1DCCNE2CDK4PRKACA
SCHEMBL9623259 0.84 CHEK1 (0.43) CHEK1MYLKROCK2
SCHEMBL9623359 0.83 GSK3A (0.45) CHEK1CCNE2CDK4CCND1CCNE1
SCHEMBL9622890 0.81 CHEK1 (0.49) CHEK1TRPM8CCNE2CDK4PRKACA
SCHEMBL29386554 0.78 PDGFRB (0.48) CHEK1HTR1DCDK4CCND1KDM4E
SCHEMBL9623119 0.78 MYLK (0.47) SLC6A4HTR1DCDK4CCND1KDM4E
SCHEMBL9622994 0.78 ROCK2 (0.45) CHEK1MYLKROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5166204-A ISOINDOLE DERIVATIVES AND SALTS THEREOF AND ANTITUMOR AGENT COMPRISING THE SAME TOYAMA CHEMICAL CO., LTD. (JP) 1992-11-24 US disclosed