SCHEMBL9623564

SCHEMBL9623564

COc1ccc2c(CCN(C)CCCN3Cc4cc5c(cc4C3=O)OCO5)csc2c1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 3/20 0.36
MAPT P10636 2/20 0.35
HCN4 Q9Y3Q4 1/20 0.35
CYP3A4 P08684 2/20 0.35
ALOX15 P16050 1/20 0.35
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624641 0.93 MTNR1A (0.39) SMPD1MAPTHCN4CYP3A4ALOX15
SCHEMBL9624428 0.90 KDM4E (0.32) MAPTHCN4KDM4EALDH1A1
SCHEMBL9624299 0.89 ITGB3 (0.34) MAPTKDM4EALDH1A1HPGD
SCHEMBL9624788 0.89 SMPD1 (0.38) SMPD1MAPTHCN4CYP3A4ALOX15
SCHEMBL9624113 0.89 HCN4 (0.44) SMPD1MAPTHCN4CYP3A4ALOX15
SCHEMBL10665062 0.87 MAPT (0.38) SMPD1MAPTHCN4CYP3A4ALOX15
SCHEMBL9625186 0.87 SMPD1 (0.34) SMPD1MAPTHCN4
SCHEMBL10663788 0.85 HCN4 (0.53) SMPD1MAPTHCN4CYP3A4ALOX15
SCHEMBL9623985 0.84 MAPT (0.44) SMPD1MAPTKDM4EALDH1A1HPGD
SCHEMBL9624301 0.84 MAPT (0.35) MAPTHCN4CYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed
EP-0269968-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-06-08 EP disclosed