SCHEMBL9624299

SCHEMBL9624299

CN(CCCN1Cc2cc3c(cc2C1=O)OCO3)CCc1csc2cc(OCC(=O)O)ccc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.34
ITGB1 P05556 1/20 0.34
ITGAV P06756 1/20 0.34
ITGA5 P08648 1/20 0.34
ITGB5 P18084 1/20 0.34
LSS P48449 1/20 0.33
PPARD Q03181 4/20 0.33
PPARA Q07869 4/20 0.33
KDM4E B2RXH2 3/20 0.32
ALDH1A1 P00352 3/20 0.32
HPGD P15428 3/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
PPARG P37231 1/20 0.32
GLA P06280 1/20 0.31
GAA P10253 1/20 0.31
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9623829 0.90 ITGB3 (0.35) ITGB3ITGB1ITGAVITGA5ITGB5
SCHEMBL9623564 0.89 SMPD1 (0.36) KDM4EALDH1A1HPGDMAPT
SCHEMBL9624306 0.89 HCN4 (0.40) ITGB3ITGB1ITGAVITGA5ITGB5
SCHEMBL9624428 0.86 KDM4E (0.32) KDM4EALDH1A1MAPTGAA
SCHEMBL9625186 0.83 SMPD1 (0.34) MAPT
SCHEMBL9624641 0.83 MTNR1A (0.39) KDM4EALDH1A1MAPT
SCHEMBL9624301 0.80 MAPT (0.35) MAPT
SCHEMBL9624076 0.80 PRKCB (0.33) MAPT
SCHEMBL9623739 0.79 CYP2A6 (0.35) MAPT
SCHEMBL9623729 0.79 AOC3 (0.35) ITGB3ITGB1ITGAVITGA5ITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed
EP-0269968-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-06-08 EP disclosed