SCHEMBL9623726

SCHEMBL9623726

Cc1ccc2[nH]cc(CCN(C)CCCN3Cc4cc(C)c(C)cc4C3=O)c2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.49
MEN1 O00255 2/20 0.49
LMNA P02545 2/20 0.49
MAPT P10636 2/20 0.49
HTT P42858 1/20 0.49
HTR2A P28223 6/20 0.43
HTR1D P28221 6/20 0.43
HTR1B P28222 5/20 0.43
HTR5A P47898 4/20 0.43
HTR1A P08908 4/20 0.43
HTR2C P28335 2/20 0.43
SLC6A4 P31645 2/20 0.43
ADRA1A P35348 2/20 0.43
ADRA2A P08913 1/20 0.43
DRD2 P14416 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
HTR1E P28566 1/20 0.43
HTR7 P34969 1/20 0.43
HRH1 P35367 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624212 0.91 SLC6A4 (0.48) KMT2AMEN1LMNAMAPTHTT
SCHEMBL9623773 0.90 BCHE (0.46) KMT2AMEN1LMNAMAPTHTT
SCHEMBL9624496 0.89 KMT2A (0.46) KMT2AMEN1LMNAMAPTHTT
SCHEMBL9624327 0.89 MAPT (0.46) KMT2AMEN1LMNAMAPTHTT
SCHEMBL9624325 0.89 HTR1A (0.52) KMT2AMEN1LMNAMAPTHTR2A
SCHEMBL9624504 0.85 HTR2A (0.43) MAPTHTR2ASLC6A4DRD2HTR6
SCHEMBL9624267 0.84 HTR1D (0.57) KMT2AMEN1LMNAMAPTHTR1D
SCHEMBL9624653 0.81 LMNA (0.46) KMT2AMEN1LMNAMAPTHTT
SCHEMBL9624529 0.81 MAPT (0.37) LMNAMAPTHTR5A
SCHEMBL9624897 0.80 HTR1A (0.52) KMT2AMEN1LMNAMAPTHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed
EP-0269968-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-06-08 EP disclosed