SCHEMBL9624504

SCHEMBL9624504

Cc1cc2c(cc1C)C(=O)N(CCCN(C)CCc1c[nH]c3c(C)cccc13)C2

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.43
MAPT P10636 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HDAC6 Q9UBN7 1/20 0.38
DRD2 P14416 2/20 0.37
SLC6A4 P31645 1/20 0.37
HTR6 P50406 1/20 0.37
SOS2 Q07890 1/20 0.37
PCSK9 Q8NBP7 1/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ALOX15 P16050 1/20 0.35
RAB9A P51151 1/20 0.35
SMPD1 P17405 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624887 0.90 HTR6 (0.45) HTR2AMAPTSMN1; SMN2NPSR1HTR6
SCHEMBL9624802 0.90 DRD2 (0.40) HTR2AMAPTSMN1; SMN2NPSR1HDAC6
SCHEMBL9623773 0.89 BCHE (0.46) HTR2AMAPTSMN1; SMN2DRD2SLC6A4
SCHEMBL9623726 0.85 KMT2A (0.49) HTR2AMAPTSMN1; SMN2DRD2SLC6A4
SCHEMBL9624212 0.83 SLC6A4 (0.48) HTR2AMAPTDRD2SLC6A4HTR6
SCHEMBL9624325 0.82 HTR1A (0.52) HTR2AMAPTSMN1; SMN2SLC6A4HTR6
SCHEMBL9624291 0.80 SMPD1 (0.36) MAPTSMN1; SMN2HDAC6DRD2HTR6
SCHEMBL9624633 0.80 SIGMAR1 (0.36) HDAC6SMPD1
SCHEMBL9624815 0.79 KDM4E (0.45) HTR2AMAPTSMN1; SMN2NPSR1DRD2
SCHEMBL9624267 0.79 HTR1D (0.57) MAPTSMN1; SMN2SLC6A4HTR6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed
EP-0269968-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-06-08 EP disclosed