SCHEMBL9628400

SCHEMBL9628400

CCCN(CCC)CC1Cc2cc(OC(=O)c3ccccc3N)ccc2O1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.39
HSD17B10 Q99714 6/20 0.39
KDM4E B2RXH2 4/20 0.39
HPGD P15428 2/20 0.39
GLA P06280 1/20 0.39
ALOX5 P09917 4/20 0.36
POLB P06746 2/20 0.35
TSHR P16473 2/20 0.35
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34
CFTR P13569 1/20 0.34
MCHR1 Q99705 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
RAB9A P51151 1/20 0.33
HIF1A Q16665 1/20 0.32
FFAR1 O14842 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9628680 0.90 KMT2A (0.42) ALDH1A1ALOX5TSHRLMNASMN1; SMN2
SCHEMBL9628391 0.79 ALDH1A1 (0.41) ALDH1A1HSD17B10KDM4EHPGDGLA
SCHEMBL10460150 0.77 ACHE (0.39) HRH3
SCHEMBL9627919 0.77 HRH3 (0.55) HRH3GABRA1GABRB2
SCHEMBL9628753 0.75 ALDH1A1 (0.42) ALDH1A1POLBSMN1; SMN2RAB9A
SCHEMBL9627815 0.73 BCHE (0.49) HPGDSMN1; SMN2RAB9A
SCHEMBL9628968 0.73 HRH3 (0.35) ALDH1A1POLBHRH3GABRA1GABRB2
SCHEMBL9627841 0.72 DRD3 (0.45) LMNAHRH3
SCHEMBL9628703 0.70 ACHE (0.45)
SCHEMBL9627868 0.70 KMT2A (0.41) ALOX5TSHRLMNASMN1; SMN2FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0281261-B1 3-AMINOMETHYL DERIVATIVES OF INDANE, INDOLINE AND DIHYDROBENZOFURANE AND DIHYDROBENZOTHIOPHENE H. LUNDBECK A/S (DK) 1992-05-06 EP disclosed
US-4946863-A CNS-affecting 6-oxy-3-aminomethyl indanes, compositions thereof, and method of treating therewith H. LUNDBECK A/S (DK) 1990-08-07 US disclosed
US-4847254-A CNS affecting 5-oxy-3-aminomethyl-dihydro-benzofurans and benzothiophenes H. LUNDBECK A/S (DK) 1989-07-11 US disclosed
EP-0281261-A2 3-Aminomethyl derivatives of indane, indoline and dihydrobenzofurane and dihydrobenzothiophene H. LUNDBECK A/S (DK) 1988-09-07 EP disclosed