SCHEMBL9628680

SCHEMBL9628680

CCCN(CCC)CC1Cc2cc(OC(=O)c3ccccc3C)ccc2O1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.42
MEN1 O00255 3/20 0.42
NPC1 O15118 3/20 0.42
CASP3 P42574 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
MAPT P10636 3/20 0.38
LMNA P02545 2/20 0.38
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
TSHR P16473 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
ALOX5 P09917 1/20 0.35
RAB9A P51151 3/20 0.35
ALDH1A1 P00352 1/20 0.35
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
MAOA P21397 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9628400 0.90 ALDH1A1 (0.39) LMNASMN1; SMN2TSHRHRH3ALOX5
SCHEMBL9627781 0.81 HRH3 (0.38) KMT2AMEN1HRH3GABRA1GABRB2
SCHEMBL9627868 0.79 KMT2A (0.41) KMT2AMEN1NPC1CASP3SENP8
SCHEMBL10460150 0.79 ACHE (0.39) HRH3
SCHEMBL9628753 0.78 ALDH1A1 (0.42) KMT2AMEN1MAPTSMN1; SMN2RAB9A
SCHEMBL9627919 0.78 HRH3 (0.55) HRH3GABRA1GABRB2
SCHEMBL9627837 0.77 KMT2A (0.41) KMT2AMEN1NPC1CASP3SENP8
SCHEMBL10460568 0.77 MGLL (0.47)
SCHEMBL9627883 0.76 ACHE (0.45) KMT2AMEN1NPC1CASP3SENP8
SCHEMBL9627815 0.74 BCHE (0.49) NPC1SMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0281261-B1 3-AMINOMETHYL DERIVATIVES OF INDANE, INDOLINE AND DIHYDROBENZOFURANE AND DIHYDROBENZOTHIOPHENE H. LUNDBECK A/S (DK) 1992-05-06 EP disclosed
US-4946863-A CNS-affecting 6-oxy-3-aminomethyl indanes, compositions thereof, and method of treating therewith H. LUNDBECK A/S (DK) 1990-08-07 US disclosed
US-4847254-A CNS affecting 5-oxy-3-aminomethyl-dihydro-benzofurans and benzothiophenes H. LUNDBECK A/S (DK) 1989-07-11 US disclosed
EP-0281261-A2 3-Aminomethyl derivatives of indane, indoline and dihydrobenzofurane and dihydrobenzothiophene H. LUNDBECK A/S (DK) 1988-09-07 EP disclosed