SCHEMBL9628968

SCHEMBL9628968

CCCN(CCC)CC1Cc2cc(OCOC(=O)C(C)(C)C)ccc2O1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.35
GABRA1 P14867 2/20 0.34
GABRB2 P47870 2/20 0.34
STING1 Q86WV6 1/20 0.33
HIF1A Q16665 1/20 0.33
FFAR1 O14842 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
PTGIR P43119 1/20 0.33
POLB P06746 1/20 0.32
GLS O94925 2/20 0.32
ITGB3 P05106 1/20 0.32
ITGA2B P08514 1/20 0.32
AKR1C4 P17516 1/20 0.31
AKR1C3 P42330 1/20 0.31
AKR1C2 P52895 1/20 0.31
AKR1C1 Q04828 1/20 0.31
PPARG P37231 3/20 0.30
PPARA Q07869 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9627781 0.88 HRH3 (0.38) HRH3GABRA1GABRB2FFAR1FFAR4
SCHEMBL9627919 0.78 HRH3 (0.55) HRH3GABRA1GABRB2GLS
SCHEMBL9628958 0.78 PPARG (0.39) FFAR1PPARGPPARA
SCHEMBL10460150 0.75 ACHE (0.39) HRH3GLS
SCHEMBL9628680 0.74 KMT2A (0.42) HRH3GABRA1GABRB2HIF1APTGIR
SCHEMBL9627841 0.73 DRD3 (0.45) HRH3
SCHEMBL9628400 0.73 ALDH1A1 (0.39) HRH3GABRA1GABRB2HIF1AFFAR1
SCHEMBL10460568 0.73 MGLL (0.47)
SCHEMBL9628753 0.73 ALDH1A1 (0.42) POLBALDH1A1
SCHEMBL9627815 0.71 BCHE (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0281261-B1 3-AMINOMETHYL DERIVATIVES OF INDANE, INDOLINE AND DIHYDROBENZOFURANE AND DIHYDROBENZOTHIOPHENE H. LUNDBECK A/S (DK) 1992-05-06 EP disclosed
US-4946863-A CNS-affecting 6-oxy-3-aminomethyl indanes, compositions thereof, and method of treating therewith H. LUNDBECK A/S (DK) 1990-08-07 US disclosed
US-4847254-A CNS affecting 5-oxy-3-aminomethyl-dihydro-benzofurans and benzothiophenes H. LUNDBECK A/S (DK) 1989-07-11 US disclosed
EP-0281261-A2 3-Aminomethyl derivatives of indane, indoline and dihydrobenzofurane and dihydrobenzothiophene H. LUNDBECK A/S (DK) 1988-09-07 EP disclosed