SCHEMBL9630558

SCHEMBL9630558

Nc1nc2ccccc2n1Cc1ccc(F)cc1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 2/20 0.75
NOD2 Q9HC29 2/20 0.75
NOD1 Q9Y239 2/20 0.75
CXCL8 P10145 1/20 0.75
SOS1 Q07889 1/20 0.75
KMT2A Q03164 2/20 0.68
RAB9A P51151 1/20 0.65
CSF1R P07333 2/20 0.63
HTT P42858 2/20 0.61
MEN1 O00255 1/20 0.61
ALDH1A1 P00352 1/20 0.61
TP53 P04637 1/20 0.61
TSHR P16473 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
NPSR1 Q6W5P4 1/20 0.61
IDO1 P14902 1/20 0.57
CYP1A2 P05177 1/20 0.57
CYP2D6 P10635 1/20 0.57
CXCR4 P61073 1/20 0.57
HTR3A P46098 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11594488 0.98 TNF (0.73) TNFNOD2NOD1CXCL8SOS1
SCHEMBL7165480 0.92 TNF (0.87) TNFNOD2NOD1CXCL8SOS1
SCHEMBL939417 0.87 TNF (0.79) TNFNOD2NOD1CXCL8SOS1
SCHEMBL7337702 0.86 NOD1 (1.00) TNFNOD2NOD1CXCL8SOS1
SCHEMBL990644 0.84 HTT (0.66) TNFNOD2NOD1CXCL8SOS1
SCHEMBL3718063 0.83 RAB9A (0.67) TNFNOD2NOD1CXCL8SOS1
SCHEMBL7530572 0.83 TNF (0.72) TNFNOD2NOD1CXCL8SOS1
SCHEMBL9537915 0.81 RAB9A (0.65) KMT2ARAB9AHTTMEN1ALDH1A1
SCHEMBL8881382 0.81 RAB9A (0.65) KMT2ARAB9AHTTMEN1ALDH1A1
SCHEMBL7168102 0.81 KMT2A (0.71) TNFNOD2NOD1CXCL8SOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5151424-A Antiallergens or antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-29 US disclosed
EP-0297661-B1 [(Bicyclic heterocyclyl)methyl and -hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-16 EP disclosed
US-5071846-A Anti-hystaminic [(bicyclic heterocyclyl) methyl and --hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1991-12-10 US disclosed
US-4988689-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1991-01-29 US disclosed
EP-0297661-A1 [(Bicyclic heterocyclyl)methyl and -hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1989-01-04 EP disclosed