SCHEMBL9635445

SCHEMBL9635445

Fc1ccc2[nH]cc(CN3CCNCC3)c2c1

nearest known ligand 0.73

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MPO P05164 8/20 0.73
SLC6A4 P31645 1/20 0.60
HTR1A P08908 4/20 0.59
GPR84 Q9NQS5 2/20 0.58
DRD2 P14416 1/20 0.57
DRD4 P21917 1/20 0.57
DRD3 P35462 1/20 0.57
HTR2A P28223 1/20 0.52
TRPM8 Q7Z2W7 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
BCHE P06276 1/20 0.51
CYP2D6 P10635 1/20 0.51
KMT2A Q03164 1/20 0.51
TSHR P16473 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5170221 0.88 MPO (0.77) MPOHTR1AGPR84DRD2DRD4
SCHEMBL13499605 0.84 MPO (1.00) MPOSLC6A4HTR1AGPR84DRD2
SCHEMBL9047205 0.84 HTR1A (0.85) MPOSLC6A4HTR1A
SCHEMBL22584707 0.83 GPR84 (0.58) MPOSLC6A4GPR84DRD2DRD4
SCHEMBL739944 0.83 HTR1A (0.79) MPOSLC6A4HTR1A
SCHEMBL14375346 0.82 MPO (0.72) MPOSLC6A4HTR1AGPR84DRD2
SCHEMBL13375737 0.80 MPO (0.69) MPOSLC6A4HTR1AGPR84DRD2
SCHEMBL17533456 0.80 HTR1A (0.62) HTR1AGPR84DRD2DRD4DRD3
SCHEMBL13374358 0.79 MPO (0.67) MPOSLC6A4HTR1AGPR84DRD2
SCHEMBL948663 0.79 CYP2D6 (0.81) SLC6A4HTR1ADRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5114949-A Treating disorders associated with 5HT uptake RHONE-POULENC SANTE (FR) 1992-05-19 US disclosed