SCHEMBL9636641

SCHEMBL9636641

COc1ccc(C(=O)N2CC3CC(C2)CN(C(C)C)C3)cc1OC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 2/20 0.53
TLR8 Q9NR97 2/20 0.53
TLR7 Q9NYK1 2/20 0.53
ALDH1A1 P00352 2/20 0.50
POLB P06746 1/20 0.50
CYP2C19 P33261 1/20 0.50
MAPK1 P28482 1/20 0.50
LMNA P02545 1/20 0.49
CHRNB2 P17787 1/20 0.48
CHRNB4 P30926 1/20 0.48
CHRNA3 P32297 1/20 0.48
CHRNA7 P36544 1/20 0.48
CHRNA4 P43681 1/20 0.48
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
ATM Q13315 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
PKM P14618 1/20 0.47
CNR2 P34972 1/20 0.47
HPGD P15428 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9636708 0.87 POLB (0.51) ALDH1A1POLBGAAPKML3MBTL1
SCHEMBL17319226 0.80 ALDH1A1 (0.61) ALDH1A1POLBCYP2C19MAPK1LMNA
SCHEMBL6336383 0.79 CHRNA7 (0.57) ALDH1A1POLBCHRNB2CHRNB4CHRNA3
SCHEMBL8711485 0.79 PAX8 (0.48) POLBCHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL9257879 0.79 CHRNB2 (0.46) ALDH1A1LMNACHRNB2CHRNB4CHRNA3
SCHEMBL6319408 0.78 CHRNB2 (0.61) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA7
Hydrochloric Acid SCHEMBL9272008 0.77 CHRNB2 (0.45) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL9264243 0.74 KMT2A (0.46) ALDH1A1POLBATMSMN1; SMN2HPGD
Hydrochloric Acid SCHEMBL9271468 0.73 KMT2A (0.45) ALDH1A1POLBATMSMN1; SMN2HPGD
SCHEMBL9636642 0.73 KDM4E (0.56) ALDH1A1MAPK1LMNAMAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110933-A Salts of 3-azabicyclo[3.3.1]nonanes as antiarrhythmic agents, and precursors thereof BOARD OF REGENTS OF OKLAHOMA STATE UNIVERSITY (US) 1992-05-05 US disclosed
US-5084572-A Cardiovascular disorders BOARD OF REGENTS OF OKLAHOMA STATE UNIVERSITY (US) 1992-01-28 US disclosed