SCHEMBL9637671

SCHEMBL9637671

CCOc1nsc(C(=O)Cl)c1Br

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
RAB9A P51151 2/20 0.32
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
HSD17B10 Q99714 1/20 0.32
THRB P10828 1/20 0.32
NPC1 O15118 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9637483 0.85 HSD17B10 (0.37) HPGDSMN1; SMN2RAB9AKDM4EGAA
SCHEMBL9637680 0.83 IKBKB (0.37) HPGDSMN1; SMN2RAB9AKDM4EGAA
SCHEMBL9637538 0.83 HPGD (0.38) HPGDSMN1; SMN2RAB9AKDM4EGAA
SCHEMBL9637450 0.82 HPGD (0.46) HPGDSMN1; SMN2RAB9AKDM4EGAA
SCHEMBL9638379 0.78 HPGD (0.33) HPGDSMN1; SMN2RAB9AKDM4EGAA
SCHEMBL9637422 0.72 L3MBTL1 (0.55) SMN1; SMN2RAB9ANPC1LMNAMAPT
SCHEMBL16986060 0.67 HPGD (0.47) HPGDSMN1; SMN2RAB9AKDM4EGAA
SCHEMBL11213214 0.66 ALDH1A1 (0.53) HPGDSMN1; SMN2RAB9AKDM4EGAA
SCHEMBL9957284 0.61 ALDH1A1 (0.39) HPGDSMN1; SMN2RAB9AKDM4EHSD17B10
SCHEMBL9638346 0.61 NPC1 (0.41) RAB9AGAANPC1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5171860-A Diamino isothiazole-1-oxides and 1,1 dioxides as gastric secretion inhibitors MERCK & CO., INC. (US) 1992-12-15 US disclosed
EP-0067436-B1 DIAMINO ISOTHIAZOLE -1-OXIDES AND -1,1-DIOXIDES AS GASTRIC SECRETION INHIBITORS MERCK & CO. INC. (US) 1986-07-23 EP disclosed
EP-0067436-A2 Diamino isothiazole -1-oxides and -1,1-dioxides as gastric secretion inhibitors MERCK & CO. INC. (US) 1982-12-22 EP disclosed